Antioxidant activity of reduced menadione in solvent solution and in model membranes

Free Radic Res. 1997 May;26(5):419-29. doi: 10.3109/10715769709084478.

Abstract

The antioxidant activity of reduced menadione was investigated and compared with that of alpha-tocopherol both in solvent solution and in large unilamellar vesicles by using azocompounds as free radical generators. The results show that: i) reduced menadione behaves as a chain-breaking antioxidant; ii) its inhibition rate constant is similar to that of alpha-tocopherol in homogeneous solution, whereas it is 4 times larger in egg yolk lecithin vesicles; iii) the stoichiometric factor is found lower than 1 in both systems, since a substantial portion of menadiol is consumed by autoxidation and does not contribute to radical trapping; iv) when both alpha-tocopherol and menadiol are present in vesicles, reduced menadione can spare alpha-tocopherol. Data presented here suggest that the reduced form of vitamin K may protect, when present, cellular membranes from free radical damage.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antioxidants / chemistry
  • Antioxidants / metabolism*
  • Antioxidants / pharmacology
  • Drug Synergism
  • Liposomes / metabolism*
  • Oxidation-Reduction
  • Phosphatidylcholines / antagonists & inhibitors
  • Phosphatidylcholines / metabolism
  • Quinones / metabolism
  • Solutions
  • Solvents / metabolism*
  • Vitamin E / metabolism
  • Vitamin E / pharmacology
  • Vitamin K / analogs & derivatives
  • Vitamin K / chemistry
  • Vitamin K / metabolism*
  • Vitamin K / pharmacology

Substances

  • Antioxidants
  • Liposomes
  • Phosphatidylcholines
  • Quinones
  • Solutions
  • Solvents
  • Vitamin K
  • Vitamin E
  • menadiol