A novel type of calcium channel sensitive to omega-agatoxin-TK in cultured rat cerebral cortical neurons

Brain Res. 1997 May 9;756(1-2):225-30. doi: 10.1016/s0006-8993(97)00202-3.

Abstract

We characterized the electrophysiological properties of calcium channels in cultured rat cerebral cortical neurons using omega-agatoxin-TK (omega-Aga-TK) by a patch-clamp technique. Two types of slowly inactivating calcium channels sensitive to omega-Aga-TK were detected. The first type showed high sensitivity to omega-Aga-TK and low recovery from the omega-Aga-TK-induced blockade during washout, corresponding to the P-type channel. The second type showed low sensitivity to omega-Aga-TK and high recovery, resembling the Q-type channel, although it was distinct from the Q-type in terms of slower inactivation kinetics. We designate this channel as Q(L)-type (long-lasting Q channel). The omega-Aga-TK-sensitive calcium channels involved in the glutamatergic synaptic transmission were also divided into two types based on the sensitivity to omega-Aga-TK and reversibility of omega-Aga-TK-induced blockade. We conclude that the Q(L)-type is a novel type of channel, and that both P-type and Q(L)-type channels play a significant role in the cerebral cortical synaptic transmission.

MeSH terms

  • Agatoxins
  • Animals
  • Calcium Channel Blockers / pharmacology*
  • Calcium Channels / drug effects*
  • Calcium Channels / physiology
  • Cells, Cultured
  • Cerebral Cortex / cytology
  • Cerebral Cortex / metabolism*
  • Electrophysiology
  • Neurons / metabolism*
  • Patch-Clamp Techniques
  • Rats / embryology
  • Rats, Wistar
  • Spider Venoms / pharmacology*
  • Synaptic Transmission / physiology

Substances

  • Agatoxins
  • Calcium Channel Blockers
  • Calcium Channels
  • Spider Venoms
  • omega-agatoxin-Aa4b