Agonist-induced activation of a non-selective ion current in glomerular endothelial cells

Kidney Int. 1997 Jul;52(1):157-64. doi: 10.1038/ki.1997.315.

Abstract

The control of intracellular calcium activity ([Ca2+]i) and membrane voltage (Vm) play an important role in regulating functions of glomerular endothelial cells (GEC). We investigated the effect of extracellular ATP on the intracellular [Ca2+]i, Vm and ion conductances in GEC. ATP (100 mumol/liter) induced a rapid increase of [Ca2+]i in GEC from 20 +/- 6 to 442 +/- 84 nmol/liter, which was followed by a sustained Ca2+ plateau of 112 +/- 29 nmol/liter. In a bath solution with a low extracellular Ca2+ concentration the ATP-induced [Ca2+]i peak was still present, but the [Ca2+]i plateau was completely prevented. In 186 experiments with the patch clamp technique the addition of ATP (1 to 100 mumol/liter) to GEC induced a transient small hyperpolarization, which was followed by a depolarization. During the ATP-induced depolarization an increase of the whole cell conductance was found. The Ca2+ ionophore A23187 (10 mumol/liter) mimicked the effect of ATP on Vm. Reduction of the extracellular Ca2+ to 1 mumol/liter itself depolarized GEC reversibly from -88 +/- 2 to -60 +/- 12 mV and increased the ATP-induced depolarization to -18 +/- 3 mV. In the absence of Na+ in the bathing solution (replacement by NMDG+) ATP induced only an attenuated depolarization and no inward current was activated. Flufenamate (100 mumol/liter), a blocker of non-selective ion channels inhibited the ATP-induced depolarization of Vm significantly by 58 +/- 13%, whereas nicardipine (10 mumol/liter) or amiloride (10 mumol/liter) had no effect. Our data indicate that the resting Vm of GEC cells is almost completely dominated by K+ conductances and that ATP activates a Ca2+ dependent non-selective ion conductance in GEC.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenosine Triphosphate / analogs & derivatives
  • Adenosine Triphosphate / pharmacology
  • Amiloride / pharmacology
  • Animals
  • Calcimycin / pharmacology
  • Calcium / analysis
  • Calcium / physiology
  • Calcium Channel Blockers / pharmacology
  • Calcium Channels / physiology*
  • Cattle
  • Cells, Cultured
  • Charybdotoxin / pharmacology
  • Chlorine / physiology
  • Endothelium / physiology
  • Flufenamic Acid / pharmacology
  • Ion Channels / physiology
  • Ion Transport*
  • Ionophores / pharmacology
  • Kidney Glomerulus / physiology*
  • Membrane Potentials
  • Nicardipine / pharmacology
  • Patch-Clamp Techniques
  • Potassium / analysis
  • Sodium / physiology
  • Thionucleotides / pharmacology
  • Uridine Triphosphate / pharmacology

Substances

  • Calcium Channel Blockers
  • Calcium Channels
  • Ion Channels
  • Ionophores
  • Thionucleotides
  • Charybdotoxin
  • Calcimycin
  • Chlorine
  • Flufenamic Acid
  • Amiloride
  • Adenosine Triphosphate
  • Sodium
  • Nicardipine
  • Potassium
  • Calcium
  • Uridine Triphosphate
  • 2-methylthio-ATP