Characterization of the interaction between the light chain of factor VIIa and tissue factor

FEBS Lett. 1997 Aug 18;413(2):359-63. doi: 10.1016/s0014-5793(97)00941-1.

Abstract

Factor VIIa (fVIIa) consists of a heavy chain (serine protease domain) and a light chain (gamma-carboxyglutamic acid (Gla)-rich and epidermal growth factor (EGF)-like domains). The light chain, primarily the first EGF-like domain, appears to provide most of the binding energy in the interaction with tissue factor (TF). The Ca2+-binding sites in the protease domain and in the first EGF-like domain influence activity and interaction with TF, but the contribution from the Ca2+-binding sites in the Gla domain has not been established. We have compared the soluble TF (sTF)-binding properties of intact fVIIa to those of a fragment comprising almost the entire light chain and a small disulphide-linked peptide from the protease domain. Half-maximal binding of fVIIa and the light chain to sTF occurred around 0.3 and 1 mM Ca2+, respectively. The Ca2+ dependence of light-chain binding indicates an influence of Ca2+ binding to the Gla domain on the interaction between fVIIa and sTF. Comparison of the sTF-binding properties of fVIIa and a truncated variant lacking the Gla domain suggests that this domain interferes with sTF association at suboptimal Ca2+ concentrations. The light chain of fVIIa associated 5-fold slower with sTF than did fVIIa at saturating Ca2+ concentrations, whereas the dissociation of its complex with sTF was at least 100-fold faster than that of fVIIa:sTF. This gave a dissociation constant of 1-2 microM for the interaction between the light chain and sTF compared to about 3 nM for the fVIIa:sTF interaction.

MeSH terms

  • 1-Carboxyglutamic Acid / metabolism
  • Animals
  • Biosensing Techniques
  • Calcium / pharmacology
  • Cells, Cultured
  • Coagulants / metabolism*
  • Cricetinae
  • Factor VIIa / genetics
  • Factor VIIa / metabolism*
  • Protein Binding
  • Recombinant Proteins / metabolism
  • Thromboplastin / metabolism*

Substances

  • Coagulants
  • Recombinant Proteins
  • 1-Carboxyglutamic Acid
  • Thromboplastin
  • Factor VIIa
  • Calcium