Peripheral mediators involved in gastric hyperemia to vagal activation by central TRH analog in rats

Am J Physiol. 1998 Jan;274(1):G170-7. doi: 10.1152/ajpgi.1998.274.1.G170.

Abstract

Mechanisms mediating the increase in gastric mucosal blood flow (GMBF) induced by the stable thyrotropin-releasing hormone (TRH) analog RX-77368 injected intracisternally at a gastric acid secretory dose (30 ng) were investigated using hydrogen gas clearance in urethan-anesthetized rats. The histamine H1 receptor antagonist pyrilamine (intravenously), capsaicin (subcutaneously, 10 days), and NG-nitro-L-arginine methyl ester (L-NAME, intracisternally) failed to impair the 150% rise in GMBF induced by intracisternal injection of RX-77368. By contrast, atropine (subcutaneously) and NG-monomethyl-L-arginine (intravenously) completely inhibited the increase in GMBF evoked by intracisternal RX-77368. L-NAME (intravenously) blocked the intracisternal RX-77368-induced increase in GMBF in capsaicin-pretreated rats, and the L-NAME effect was reversed by intravenous L- but not D-arginine. These findings indicate that vagal efferent activation induced by TRH analog injected intracisternally at a gastric acid secretory dose increases GMBF through atropine-sensitive mechanisms stimulating L-arginine-nitric oxide pathways, whereas H1 receptors and capsaicin-sensitive afferent fibers do not play a role.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Arginine / pharmacology
  • Atropine / pharmacology
  • Blood Pressure / drug effects
  • Capsaicin / pharmacology
  • Cisterna Magna / drug effects
  • Cisterna Magna / physiology*
  • Electric Stimulation
  • Gastric Acid / metabolism*
  • Gastric Mucosa / blood supply*
  • Gastric Mucosa / drug effects
  • Gastric Mucosa / innervation
  • Hyperemia*
  • Male
  • NG-Nitroarginine Methyl Ester / pharmacology
  • Pyrrolidonecarboxylic Acid / analogs & derivatives
  • Rats
  • Rats, Sprague-Dawley
  • Stereoisomerism
  • Stereotaxic Techniques
  • Thyrotropin-Releasing Hormone / administration & dosage
  • Thyrotropin-Releasing Hormone / analogs & derivatives*
  • Thyrotropin-Releasing Hormone / pharmacology
  • Vagus Nerve / drug effects
  • Vagus Nerve / physiology*
  • Vascular Resistance / drug effects

Substances

  • Thyrotropin-Releasing Hormone
  • L-pyroglutamyl-L-histidyl-3,3-dimethylprolinamide
  • Atropine
  • Arginine
  • Capsaicin
  • Pyrrolidonecarboxylic Acid
  • NG-Nitroarginine Methyl Ester