Indium-111-pentetreotide in Graves' disease

J Nucl Med. 1998 Mar;39(3):533-6.

Abstract

Thyroidal and orbital lymphocytic infiltration in Graves' disease, as well as identification of somatostatin receptors on lymphocytes, has provided a rationale for receptor imaging with the radiolabeled somatostatin analog pentetreotide. Recently, we demonstrated that in contrast to controls, Graves' patients showed markedly increased orbital accumulation of pentetreotide. Longitudinal and follow-up data are presented here.

Methods: In 20 (16 hyperthyroid) Graves' patients with active eye disease, planar (thyroid) and SPECT (orbit) images were performed 4 and 24 hr after injection of 111In-pentetreotide (222 MBq) before and 3 mo after starting antithyroid and combined steroid and orbital radiotherapy.

Results: Thyroidal uptake decreased during methimazole treatment (4 hr postinjection, median: hyperthyroid 989 counts/pixel/MBq injected activity, euthyroid 253 counts, p = 0.001; 24 hr, 437 versus 95 counts/pixel/MBq, p = 0.005). Fourteen patients (70%) responded to steroid and radiotherapy. The pentetreotide orbit-to-brain ratio decreased markedly after completion of therapy (4 hr: 25 before versus 6.2 after therapy, p = 0.0003; 24 hr: 9.6 versus 2.7, p = 0.003). A high pretreatment ratio correlated with a response to therapy (p = 0.001: in 14 of 16 patients with a ratio > 10, 4 hr postinjection, ophthalmopathy improved; positive predictive value: 90%; median activity score before 6 versus 2 after therapy, p = 0.0001) in contrast to none of the four cases with a ratio less than 10 (score 5 versus 4, p = 0.08).

Conclusion: Pentetreotide scans may be regarded as a semiobjective tool in the evaluation of Graves' disease, both at initial stages as well as during treatment.

MeSH terms

  • Anti-Inflammatory Agents / therapeutic use
  • Antithyroid Agents / therapeutic use
  • Cobalt Radioisotopes / therapeutic use
  • Female
  • Follow-Up Studies
  • Graves Disease / diagnostic imaging*
  • Graves Disease / drug therapy
  • Graves Disease / epidemiology
  • Graves Disease / radiotherapy
  • Humans
  • Indium Radioisotopes*
  • Longitudinal Studies
  • Male
  • Methimazole / therapeutic use
  • Middle Aged
  • Predictive Value of Tests
  • Prednisolone / therapeutic use
  • Prospective Studies
  • Radioisotope Teletherapy
  • Radiopharmaceuticals*
  • Receptors, Somatostatin / analysis*
  • Sensitivity and Specificity
  • Somatostatin / analogs & derivatives*
  • Tomography, Emission-Computed, Single-Photon

Substances

  • Anti-Inflammatory Agents
  • Antithyroid Agents
  • Cobalt Radioisotopes
  • Indium Radioisotopes
  • Radiopharmaceuticals
  • Receptors, Somatostatin
  • Somatostatin
  • Methimazole
  • Prednisolone
  • pentetreotide