Characterization of a mouse monoclonal IgG3 antibody to the tumor-associated globo H structure produced by immunization with a synthetic glycoconjugate

Glycoconj J. 1998 Mar;15(3):243-9. doi: 10.1023/a:1006992911709.

Abstract

Globo H (Fuc alpha1 --> 2Galbeta1 --> 3GalNAcbeta1 --> 3Gal alpha1 --> 4Galbeta1 --> 4Glc) is a carbohydrate structure that shows enhanced expression in many human carcinomas. From mice immunized with a globo H-KLH (keyhole limpet hemocyanin) synthetic conjugate an IgG3 monoclonal antibody (mAb VK-9) was derived that recognizes the globo H structure. Serological analysis showed that the minimal structure recognized by this mAb was the tetrasaccharide sequence Fuc alpha1 --> 2Galbeta1 --> 3GalNAcbeta1 --> 3Gal. An isomeric structure with an internal alphaGalNAc linkage was also recognized but less efficiently. mAb VK-9 did not react with many related structures, such as galactosylgloboside, globoside, H type 1, H type 2 blood group structures or fucosyl-gangliotetraosyl ceramide, but did react weakly with globo A ceramide. Not only did mAb VK-9 react with carbohydrate-protein conjugates but it could also recognize globo H-ceramide and human tumor cells expressing globo H. These results suggest that globo H-KLH could be explored as a vaccine in the treatment of carcinoma patients.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Antibodies, Monoclonal / immunology*
  • Antibody Specificity
  • Antigens, Tumor-Associated, Carbohydrate / chemistry*
  • Cancer Vaccines / chemistry
  • Cancer Vaccines / isolation & purification
  • Carbohydrate Sequence
  • Female
  • Glycoconjugates / chemistry
  • Glycoconjugates / immunology
  • Hemocyanins / immunology
  • Humans
  • Immunization
  • Immunoglobulin G / immunology*
  • Mice
  • Molecular Sequence Data
  • Vaccines, Conjugate / chemistry
  • Vaccines, Conjugate / isolation & purification

Substances

  • Antibodies, Monoclonal
  • Antigens, Tumor-Associated, Carbohydrate
  • Cancer Vaccines
  • Glycoconjugates
  • Immunoglobulin G
  • Vaccines, Conjugate
  • Hemocyanins
  • keyhole-limpet hemocyanin