Change of level and expression of endothelin-1 in the lungs of rats with hypoxic pulmonary hypertension

Chin Med J (Engl). 1997 Feb;110(2):104-8.

Abstract

Objective: To determine whether mRNA for endothelin-1 was present and changed in the lungs of rats exposed to chronic hypoxia.

Methods: cRNA probes for rat ET-1 and c-fos were labelled by in vitro transcription with digoxigenin-UTP for in situ hybridization. Endothelin-1 like immunoreactivity (ET-1-LI) in plasma as well as in lung homogenate was measured by radioimmunoassay.

Results: The vascular endothelial cells of pulmonary arteries and the bronchiolar epithelial cells were strongly positive for the ET-1 probe. The perivascular and peribronchiolar smooth muscle were positive for the c-fos probe, primarily. There was little expression of ET-1 and c-fos in the rat lungs in controls. There was significant increase of ET-1-LI levels in rats exposed to hypoxia for 3 weeks, the concentration ET-1-LI in venous samples was 3.85 +/- 1.52 ng/L (P < 0.05 as compared with the control groups), in arterial sample was 4.72 +/- 1.66 ng/L (P < 0.05) and in lung was 2.06 +/- 0.68 ng/g wet lung weight (P < 0.05).

Conclusions: Chronic hypoxia elevated the mean pulmonary arterial pressure, caused vessel remodelling and the right ventricular hypertrophy. These changes were accompanied by an increase of ET-1 in plasma and lung homogenate. The expression and production of ET-1 were localized to endothelium and airway epithelium in the lungs.

MeSH terms

  • Animals
  • Endothelin-1 / biosynthesis
  • Endothelin-1 / metabolism*
  • Gene Expression
  • Hypertension, Pulmonary / etiology
  • Hypertension, Pulmonary / metabolism*
  • Hypoxia / complications*
  • Lung / metabolism*
  • Male
  • Proto-Oncogene Proteins c-fos / biosynthesis
  • RNA, Messenger / biosynthesis
  • Rats
  • Rats, Wistar

Substances

  • Endothelin-1
  • Proto-Oncogene Proteins c-fos
  • RNA, Messenger