Regulation of amiloride-sensitive sodium absorption in murine airway epithelium by C-type natriuretic peptide

Am J Physiol. 1998 Jun;274(6):L990-6. doi: 10.1152/ajplung.1998.274.6.L990.

Abstract

We have previously shown that C-type natriuretic peptide (CNP), a guanylate cyclase agonist, can stimulate cystic fibrosis transmembrane conductance regulator (CFTR)-mediated chloride secretion in murine airway epithelial cells via protein kinase (PK) A activation through the inhibition of cGMP-inhibited phosphodiesterases. In this paper, we show that CNP is also capable of reducing amiloride-sensitive sodium absorption in murine airway epithelium through a cGMP-dependent mechanism that is separate from the CFTR regulatory signaling pathway. Both murine tracheal and nasal tissues exhibit sensitivity to amiloride-sensitive sodium regulation by exogenously added CNP. CNP depolarized the nasal transepithelial potential difference by 6.3 +/- 0.5 mV, whereas the cGMP-inhibited phosphodiesterase inhibitor milrinone actually hyperpolarized the nasal transepithelial potential difference by 2.0 +/- 1.2 mV in mice homozygous for a CFTR stop mutation [CFTR(-/-)]. Inhibition of guanylate cyclase activity and PKG activity in normal mice resulted in an increase in amiloride-sensitive sodium absorption, suggesting that tonic regulation of amiloride-sensitive sodium absorption is in part due to basal cGMP levels and PKG activity.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 8-Bromo Cyclic Adenosine Monophosphate / pharmacology
  • Absorption
  • Amiloride / pharmacology*
  • Animals
  • Biological Transport / drug effects
  • Cyclic AMP-Dependent Protein Kinases / metabolism
  • Cyclic GMP / pharmacology
  • Cystic Fibrosis Transmembrane Conductance Regulator / genetics
  • Epithelium / metabolism
  • Membrane Potentials
  • Mice
  • Milrinone
  • Mutation
  • Nasal Mucosa / drug effects
  • Nasal Mucosa / metabolism*
  • Natriuretic Peptide, C-Type
  • Phosphodiesterase Inhibitors / pharmacology
  • Proteins / pharmacology*
  • Pyridones / pharmacology
  • Sodium / metabolism*
  • Trachea / drug effects
  • Trachea / metabolism*

Substances

  • Phosphodiesterase Inhibitors
  • Proteins
  • Pyridones
  • Cystic Fibrosis Transmembrane Conductance Regulator
  • Natriuretic Peptide, C-Type
  • 8-Bromo Cyclic Adenosine Monophosphate
  • Amiloride
  • Sodium
  • Cyclic AMP-Dependent Protein Kinases
  • Cyclic GMP
  • Milrinone