Transforming growth factor-beta receptor expression on human skin fibroblasts: dimeric complex formation of type I and type II receptors and identification of glycosyl phosphatidylinositol-anchored transforming growth factor-beta binding proteins

J Cell Physiol. 1998 Sep;176(3):553-64. doi: 10.1002/(SICI)1097-4652(199809)176:3<553::AID-JCP12>3.0.CO;2-0.

Abstract

Fibroblasts play a critical role in wound repair and in the development of fibrotic diseases, and transforming growth factor-beta (TGF-beta) has been shown to profoundly modulate fibroblast function. However, there is limited information on the TGF-beta receptor types, isoform specificity, and complex formation in skin fibroblasts. Here, we report that normal adult human skin fibroblasts display two isoform-specific, cell surface glycosyl phosphatidylinositol (GPI)-anchored, TGF-beta binding proteins in addition to the type I, II, and III TGF-beta receptors. The identities of these proteins are confirmed on the basis of their affinity for TGF-beta isoforms, immunoprecipitation with specific antireceptor antibodies, and other biochemical analyses. Immunoprecipitation results also indicated oligomeric complex formation between type I and II and between type II and III TGF-beta receptors. Furthermore, by using affinity labeling and two-dimensional electrophoresis, we demonstrate the occurrence of type I and II heterodimers and type I homodimers of TGF-beta receptors on these cells. Because the type I receptor does not bind TGF-beta in the absence of type II receptor, these results indicate that one molecule of TGF-beta induces the formation of a heterooligomeric complex containing more than one molecule each of type I and II TGF-beta receptors on these cells. These cells respond to TGF-beta by markedly down-regulating all five binding proteins and by potently augmenting DNA synthesis. These results allow the expansion of the proposed heteromeric TGF-beta receptor signaling paradigm using mutant cells that are unresponsive to TGF-beta and cell lines that have been transfected to overexpress these receptors, to include normal TGF-beta-responsive cells. In addition, the definition of TGF-beta receptor profiles in human skin fibroblasts provides important information for studying their alterations in these cells in various skin diseases.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Activin Receptors, Type I*
  • Antibodies
  • Antioxidants / pharmacology
  • Cells, Cultured
  • Dimerization
  • Dithiothreitol / analogs & derivatives
  • Dithiothreitol / pharmacology
  • Electrophoresis, Gel, Two-Dimensional
  • Fibroblasts / chemistry
  • Fibroblasts / cytology
  • Glycosylphosphatidylinositols / analysis*
  • Homeostasis / physiology
  • Humans
  • Isomerism
  • Phosphatidylinositol Diacylglycerol-Lyase
  • Precipitin Tests
  • Protein Binding / drug effects
  • Protein Serine-Threonine Kinases / biosynthesis*
  • Protein Serine-Threonine Kinases / chemistry
  • Protein Serine-Threonine Kinases / immunology
  • Receptor, Transforming Growth Factor-beta Type I
  • Receptor, Transforming Growth Factor-beta Type II
  • Receptors, Transforming Growth Factor beta / biosynthesis*
  • Receptors, Transforming Growth Factor beta / chemistry
  • Receptors, Transforming Growth Factor beta / immunology
  • Signal Transduction / physiology
  • Skin / chemistry
  • Skin / cytology*
  • Transfection
  • Transforming Growth Factor beta / chemistry
  • Transforming Growth Factor beta / metabolism
  • Type C Phospholipases / pharmacology

Substances

  • Antibodies
  • Antioxidants
  • Glycosylphosphatidylinositols
  • Receptors, Transforming Growth Factor beta
  • Transforming Growth Factor beta
  • dithiothreitol tetraacetate
  • Protein Serine-Threonine Kinases
  • Activin Receptors, Type I
  • Receptor, Transforming Growth Factor-beta Type I
  • Receptor, Transforming Growth Factor-beta Type II
  • Type C Phospholipases
  • Phosphatidylinositol Diacylglycerol-Lyase
  • Dithiothreitol