Evidence for ryanodine receptors in Schistosoma mansoni

Biochem Pharmacol. 1998 Oct 15;56(8):997-1003. doi: 10.1016/s0006-2952(98)00219-6.

Abstract

The present study investigated the presence of ryanodine receptors in the trematode Schistosoma mansoni. [3H]Ryanodine specific binding sites were found in the four subcellular fractions of S. mansoni; however, more binding sites were recovered in the heterogeneous fraction P1 and the microsomal fraction P4, as was thapsigargin-sensitive (Ca2+-Mg2+)ATPase activity, marking the sarco/endoplasmic reticulum calcium ATPase (SERCA) pumps. This binding had an equilibrium dissociation constant (Kd) in the nanomolar range, an apparent maximal number of receptors (Bmax) of about 80 fmol/mg of protein, and was modulated by ions (Ca2+, Mg2+) and some pharmacological tools such as caffeine. Ryanodine was able to accelerate the rate of 45Ca2+ release from actively loaded vesicles, and also to induce a transient contraction of the whole worm. We conclude that ryanodine-sensitive Ca2+ release channels are present in S. mansoni, with properties very similar to the ones present in higher animals.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Calcium / metabolism*
  • Calcium Channels / drug effects*
  • Male
  • Muscle Contraction / drug effects
  • Rats
  • Ryanodine / pharmacology*
  • Ryanodine Receptor Calcium Release Channel / analysis*
  • Schistosoma mansoni / chemistry*

Substances

  • Calcium Channels
  • Ryanodine Receptor Calcium Release Channel
  • Ryanodine
  • Calcium