Perioperative pharmacokinetics of transdermal fentanyl in elderly and young adult patients

Br J Anaesth. 1998 Aug;81(2):152-4. doi: 10.1093/bja/81.2.152.

Abstract

The perioperative pharmacokinetics of transdermally-delivered fentanyl were compared in 10 young adult (mean [range] age 32.7, [25-38] yr) and eight elderly (mean [range] age 73.7 [64-82] yr) patients following abdominal surgery. Transdermal fentanyl patches designed to release 50 micrograms h-1 were applied 2 h preoperatively and left in place for 72 h. Plasma fentanyl concentrations were measured by radioimmunoassay during patch application and for 30 h after patch removal. The mean half-time (time for plasma concentrations to double after patch application) was 4.2 h in the younger group and 11.1 h in the elderly group (P < 0.005). Mean maximum plasma concentrations were 1.9 ng ml-1 and 1.5 ng ml-1 in the younger and elderly groups respectively (ns). There were no differences in the time at which maximum plasma concentrations occurred (tmax), elimination half-life after patch removal, or AUC(0-infinity).

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Abdomen / surgery
  • Administration, Cutaneous
  • Adult
  • Age Factors
  • Aged
  • Aged, 80 and over
  • Analgesics, Opioid / blood*
  • Analgesics, Opioid / pharmacokinetics
  • Anesthesia, General
  • Female
  • Fentanyl / blood*
  • Fentanyl / pharmacokinetics
  • Half-Life
  • Humans
  • Male
  • Middle Aged
  • Radioimmunoassay

Substances

  • Analgesics, Opioid
  • Fentanyl