Organometallic photonucleases: a novel class of DNA-cleaving agents

Bioorg Med Chem Lett. 1998 Apr 7;8(7):871-4. doi: 10.1016/s0960-894x(98)00127-9.

Abstract

The first demonstration of DNA cleavage by an organic radical generated via homolysis of a metal-alkyl bond in a Cp-metal complex is presented. Irradiation of CpW(CO)3CH3 (1.5 molecules/base pair) produced methyl radical, giving single-strand cleavage of pBR322 DNA. This process was inhibited by the general radical trap cysteine and by TEMPO, which traps carbon radicals but not oxygen-centered radicals.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cyclic N-Oxides
  • Cysteine
  • DNA / chemistry*
  • Deoxyribonucleases*
  • Free Radicals
  • Organometallic Compounds / chemical synthesis
  • Organometallic Compounds / chemistry*
  • Photolysis
  • Plasmids / chemistry*

Substances

  • Cyclic N-Oxides
  • Free Radicals
  • Organometallic Compounds
  • DNA
  • Deoxyribonucleases
  • Cysteine
  • TEMPO