Synthesis and ESR study of new dihydroxamic acid siderophores S as scavengers of hydroxyl radicals

Bioorg Med Chem Lett. 1998 Feb 3;8(3):227-32. doi: 10.1016/s0960-894x(97)10219-0.

Abstract

Five new dihydroxamic acid ligands (L) (8, 10a, 10b, 10c and 13) have been synthesised and characterised as potential chelating agents for iron (Fe3+). The log stability constants of Fe2L3 and FeL+ from Fe3+ and L2- have been estimated to be log beta = 61.96 and log beta 1 = 22.8 respectively. The ability of these compounds to scavenge hydroxyl radicals (oOH) responsible for cell damage have been studied by esr spectroscopy.

MeSH terms

  • Electron Spin Resonance Spectroscopy
  • Free Radical Scavengers / chemical synthesis*
  • Free Radical Scavengers / chemistry
  • Free Radical Scavengers / pharmacology
  • Hydroxamic Acids / chemical synthesis*
  • Hydroxamic Acids / chemistry
  • Hydroxamic Acids / pharmacology
  • Hydroxyl Radical / chemistry*
  • Magnetic Resonance Spectroscopy
  • Siderophores / chemical synthesis*
  • Siderophores / chemistry
  • Siderophores / pharmacology

Substances

  • Free Radical Scavengers
  • Hydroxamic Acids
  • Siderophores
  • Hydroxyl Radical