Synthesis and biological activity of novel thiazolidinediones

Bioorg Med Chem Lett. 1998 Oct 6;8(19):2725-30. doi: 10.1016/s0960-894x(98)00485-5.

Abstract

Novel compounds having a dual pharmacophore were synthesised and evaluated for their insulin sensitiser and anti-inflammatory properties in different animal models.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Inflammatory Agents, Non-Steroidal / chemical synthesis*
  • Anti-Inflammatory Agents, Non-Steroidal / pharmacology*
  • Blood Glucose / drug effects
  • Butanones / pharmacology
  • Chromans / pharmacology
  • Edema / drug therapy
  • Female
  • Hypoglycemic Agents / chemical synthesis*
  • Hypoglycemic Agents / pharmacology*
  • Male
  • Mice
  • Nabumetone
  • Rats
  • Rats, Wistar
  • Structure-Activity Relationship
  • Thiazoles / chemical synthesis*
  • Thiazoles / pharmacology*
  • Thiazolidinediones*
  • Troglitazone

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • Blood Glucose
  • Butanones
  • Chromans
  • Hypoglycemic Agents
  • Thiazoles
  • Thiazolidinediones
  • Troglitazone
  • Nabumetone
  • netoglitazone