Anthelmintic beta-hydroxyketoamides (BKAs)

Bioorg Med Chem Lett. 1998 Dec 1;8(23):3317-20. doi: 10.1016/s0960-894x(98)00588-5.

Abstract

We have prepared several anthelmintic coumarins based on the beta-hydroxyketoamide (BKA) template and have shown that this template remains valid over a wide range of changes to the coumarin moiety allowing for the inclusion of carbocyclic, bicyclic, and heterocyclic rings.

MeSH terms

  • Animals
  • Anthelmintics / chemical synthesis*
  • Anthelmintics / pharmacology
  • Coumarins / chemical synthesis*
  • Coumarins / pharmacology
  • Gerbillinae

Substances

  • Anthelmintics
  • Coumarins