Cloning and evaluation of the role of rat GALR-2, a novel subtype of galanin receptor, in the control of pain perception

Ann N Y Acad Sci. 1998 Dec 21:863:108-19. doi: 10.1111/j.1749-6632.1998.tb10688.x.

Abstract

We have identified a novel subtype of galanin receptor (GALR-2) in rat dorsal root ganglia and spinal cord. The open reading frame of GALR-2 is 1116 nucleotides long, encoding a protein of 372 amino acids with a theoretical molecular mass of 40.7 kD. Membranes prepared from stable pools of 293 cells expressing GALR-2, but not wild-type 293 cells, demonstrated high affinity galanin binding sites. Rat galanin and galanin-related peptides M40, C7, M15, and galanin effectively competed for binding; peptide C7 demonstrated a lower affinity for rGALR-2, and all these peptides were agonists at rGALR-2 when assessed on a microphysiometer. Studies on the expression of GALR-2 in various tissues by Northern and in situ hybridization analyses suggest a low abundance but wide distribution of GALR-2 mRNA, including several discrete areas in brain and spinal cord and a high abundance in the dorsal root ganglia.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Base Sequence
  • Cloning, Molecular
  • Ganglia, Spinal / physiology
  • In Situ Hybridization
  • Male
  • Molecular Sequence Data
  • Organ Specificity
  • Pain / physiopathology*
  • RNA, Messenger / analysis
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, Galanin
  • Receptors, Neuropeptide / physiology*
  • Spinal Cord / physiology

Substances

  • RNA, Messenger
  • Receptors, Galanin
  • Receptors, Neuropeptide