Baraldi PG - Search Results

1

Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists.

Baraldi PG, Cacciari B, Romagnoli R, Spalluto G, Klotz KN, Leung E, Varani K, Gessi S, Merighi S, Borea PA. Baraldi PG, et al. J Med Chem. 1999 Nov 4;42(22):4473-8. doi: 10.1021/jm991114s. J Med Chem. 1999. PMID: 10579811 No abstract available.

2

7-Substituted 5-amino-2-(2-furyl)pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonists: a study on the importance of modifications at the side chain on the activity and solubility.

Baraldi PG, Cacciari B, Romagnoli R, Spalluto G, Monopoli A, Ongini E, Varani K, Borea PA. Baraldi PG, et al. J Med Chem. 2002 Jan 3;45(1):115-26. doi: 10.1021/jm010924c. J Med Chem. 2002. PMID: 11754583

3

Synthesis, biological activity, and molecular modeling investigation of new pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as human A(3) adenosine receptor antagonists.

Baraldi PG, Cacciari B, Moro S, Spalluto G, Pastorin G, Da Ros T, Klotz KN, Varani K, Gessi S, Borea PA. Baraldi PG, et al. J Med Chem. 2002 Feb 14;45(4):770-80. doi: 10.1021/jm0109614. J Med Chem. 2002. PMID: 11831890

4

Synthesis, biological properties, and molecular modeling investigation of the first potent, selective, and water-soluble human A(3) adenosine receptor antagonist.

Maconi A, Pastorin G, Da Ros T, Spalluto G, Gao ZG, Jacobson KA, Baraldi PG, Cacciari B, Varani K, Moro S, Borea PA. Maconi A, et al. Among authors: baraldi pg. J Med Chem. 2002 Aug 15;45(17):3579-82. doi: 10.1021/jm020974x. J Med Chem. 2002. PMID: 12166930 Free PMC article.

5

Pyrazolo-triazolo-pyrimidine derivatives as adenosine receptor antagonists: a possible template for adenosine receptor subtypes?

Baraldi PG, Cacciari B, Borean PA, Varanin K, Pastorin G, Da Ros T, Tabrizi MA, Fruttarolo F, Spalluto G. Baraldi PG, et al. Curr Pharm Des. 2002;8(26):2299-332. doi: 10.2174/1381612023392838. Curr Pharm Des. 2002. PMID: 12369947 Review.

6

Synthesis and biological effects of novel 2-amino-3-naphthoylthiophenes as allosteric enhancers of the A1 adenosine receptor.

Baraldi PG, Romagnoli R, Pavani MG, Nuñez Mdel C, Tabrizi MA, Shryock JC, Leung E, Moorman AR, Uluoglu C, Iannotta V, Merighi S, Borea PA. Baraldi PG, et al. J Med Chem. 2003 Feb 27;46(5):794-809. doi: 10.1021/jm0210212. J Med Chem. 2003. PMID: 12593659

7

Design, synthesis, and biological evaluation of C9- and C2-substituted pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as new A2A and A3 adenosine receptors antagonists.

Baraldi PG, Fruttarolo F, Tabrizi MA, Preti D, Romagnoli R, El-Kashef H, Moorman A, Varani K, Gessi S, Merighi S, Borea PA. Baraldi PG, et al. J Med Chem. 2003 Mar 27;46(7):1229-41. doi: 10.1021/jm021023m. J Med Chem. 2003. PMID: 12646033

8

Recent developments in the field of A2A and A3 adenosine receptor antagonists.

Baraldi PG, Tabrizi MA, Bovero A, Avitabile B, Preti D, Fruttarolo F, Romagnoli R, Varani K, Borea PA. Baraldi PG, et al. Eur J Med Chem. 2003 Apr;38(4):367-82. doi: 10.1016/s0223-5234(03)00042-4. Eur J Med Chem. 2003. PMID: 12750024

9

New strategies for the synthesis of A3 adenosine receptor antagonists.

Baraldi PG, Bovero A, Fruttarolo F, Romagnoli R, Tabrizi MA, Preti D, Varani K, Borea PA, Moorman AR. Baraldi PG, et al. Bioorg Med Chem. 2003 Sep 15;11(19):4161-9. doi: 10.1016/s0968-0896(03)00484-x. Bioorg Med Chem. 2003. PMID: 12951147

10

Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as adenosine receptor antagonists. Influence of the N5 substituent on the affinity at the human A 3 and A 2B adenosine receptor subtypes: a molecular modeling investigation.

Pastorin G, Da Ros T, Spalluto G, Deflorian F, Moro S, Cacciari B, Baraldi PG, Gessi S, Varani K, Borea PA. Pastorin G, et al. Among authors: baraldi pg. J Med Chem. 2003 Sep 25;46(20):4287-96. doi: 10.1021/jm030852k. J Med Chem. 2003. PMID: 13678407

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

247 results

Search Page

Filters