Yang YT - Search Results

1

Potent antagonists of gonadotropin releasing hormone receptors derived from quinolone-6-carboxamides.

Walsh TF, Toupence RB, Young JR, Huang SX, Ujjainwalla F, DeVita RJ, Goulet MT, Wyvratt MJ Jr, Fisher MH, Lo JL, Ren N, Yudkovitz JB, Yang YT, Cheng K, Smith RG. Walsh TF, et al. Among authors: yang yt. Bioorg Med Chem Lett. 2000 Mar 6;10(5):443-7. doi: 10.1016/s0960-894x(00)00024-x. Bioorg Med Chem Lett. 2000. PMID: 10743944

2

Identification and initial structure-activity relationships of a novel non-peptide quinolone GnRH receptor antagonist.

DeVita RJ, Hollings DD, Goulet MT, Wyvratt MJ, Fisher MH, Lo JL, Yang YT, Cheng K, Smith RG. DeVita RJ, et al. Among authors: yang yt. Bioorg Med Chem Lett. 1999 Sep 6;9(17):2615-20. doi: 10.1016/s0960-894x(99)00446-1. Bioorg Med Chem Lett. 1999. PMID: 10498220

3

Investigation of the 4-O-alkylamine substituent of non-peptide quinolone GnRH receptor antagonists.

DeVita RJ, Goulet MT, Wyvratt MJ, Fisher MH, Lo JL, Yang YT, Cheng K, Smith RG. DeVita RJ, et al. Among authors: yang yt. Bioorg Med Chem Lett. 1999 Sep 6;9(17):2621-4. doi: 10.1016/s0960-894x(99)00447-3. Bioorg Med Chem Lett. 1999. PMID: 10498221

4

Quinolones as gonadotropin releasing hormone (GnRH) antagonists: simultaneous optimization of the C(3)-aryl and C(6)-substituents.

Young JR, Huang SX, Chen I, Walsh TF, DeVita RJ, Wyvratt MJ Jr, Goulet MT, Ren N, Lo J, Yang YT, Yudkovitz JB, Cheng K, Smith RG. Young JR, et al. Among authors: yang yt. Bioorg Med Chem Lett. 2000 Aug 7;10(15):1723-7. doi: 10.1016/s0960-894x(00)00318-8. Bioorg Med Chem Lett. 2000. PMID: 10937733

5

Initial structure-activity relationship of a novel class of nonpeptidyl GnRH receptor antagonists: 2-arylindoles.

Chu L, Hutchins JE, Weber AE, Lo JL, Yang YT, Cheng K, Smith RG, Fisher MH, Wyvratt MJ, Goulet MT. Chu L, et al. Among authors: yang yt. Bioorg Med Chem Lett. 2001 Feb 26;11(4):509-13. doi: 10.1016/s0960-894x(00)00707-1. Bioorg Med Chem Lett. 2001. PMID: 11229759

6

SAR studies of novel 5-substituted 2-arylindoles as nonpeptidyl GnRH receptor antagonists.

Chu L, Lo JL, Yang YT, Cheng K, Smith RG, Fisher MH, Wyvratt MJ, Goulet MT. Chu L, et al. Among authors: yang yt. Bioorg Med Chem Lett. 2001 Feb 26;11(4):515-7. doi: 10.1016/s0960-894x(00)00708-3. Bioorg Med Chem Lett. 2001. PMID: 11229760

7

A potent, nonpeptidyl 1H-quinolone antagonist for the gonadotropin-releasing hormone receptor.

DeVita RJ, Walsh TF, Young JR, Jiang J, Ujjainwalla F, Toupence RB, Parikh M, Huang SX, Fair JA, Goulet MT, Wyvratt MJ, Lo JL, Ren N, Yudkovitz JB, Yang YT, Cheng K, Cui J, Mount G, Rohrer SP, Schaeffer JM, Rhodes L, Drisko JE, McGowan E, MacIntyre DE, Vincent S, Carlin JR, Cameron J, Smith RG. DeVita RJ, et al. Among authors: yang yt. J Med Chem. 2001 Mar 15;44(6):917-22. doi: 10.1021/jm000275p. J Med Chem. 2001. PMID: 11300873

8

2-(3,5-Dimethylphenyl)tryptamine derivatives that bind to the GnRH receptor.

Lin P, Marino D, Lo JL, Yang YT, Cheng K, Smith RG, Fisher MH, Wyvratt MJ, Goulet MT. Lin P, et al. Among authors: yang yt. Bioorg Med Chem Lett. 2001 Apr 23;11(8):1073-6. doi: 10.1016/s0960-894x(01)00134-2. Bioorg Med Chem Lett. 2001. PMID: 11327593

9

Heterocyclic derivatives of 2-(3,5-dimethylphenyl)tryptamine as GnRH receptor antagonists.

Lin P, Parikh M, Lo JL, Yang YT, Cheng K, Smith RG, Fisher MH, Wyvratt MJ, Goulet MT. Lin P, et al. Among authors: yang yt. Bioorg Med Chem Lett. 2001 Apr 23;11(8):1077-80. doi: 10.1016/s0960-894x(01)00133-0. Bioorg Med Chem Lett. 2001. PMID: 11327594

10

Substituted indole-5-carboxamides and -acetamides as potent nonpeptide GnRH receptor antagonists.

Ashton WT, Sisco RM, Yang YT, Lo JL, Yudkovitz JB, Cheng K, Goulet MT. Ashton WT, et al. Among authors: yang yt. Bioorg Med Chem Lett. 2001 Jul 9;11(13):1723-6. doi: 10.1016/s0960-894x(01)00274-8. Bioorg Med Chem Lett. 2001. PMID: 11425546

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