Discovery of 1-(Phenylsulfonyl)-1,2,3,4-tetrahydroquinoline Derivative as Orally Bioavailable and Safe RORγt Inverse Agonists for Potential Treatment of Rheumatoid Arthritis.
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J Med Chem. 2024 Nov 15. doi: 10.1021/acs.jmedchem.4c01727. Online ahead of print.
J Med Chem. 2024.
PMID: 39546350