Menge WM - Search Results

1

Synthesis and use of FSCPX, an irreversible adenosine A1 antagonist, as a 'receptor knock-down' tool.

van Muijlwijk-Koezen JE, Timmerman H, van der Sluis RP, van de Stolpe AC, Menge WM, Beukers MW, van der Graaf PH, de Groote M, IJzerman AP. van Muijlwijk-Koezen JE, et al. Among authors: menge wm. Bioorg Med Chem Lett. 2001 Mar 26;11(6):815-8. doi: 10.1016/s0960-894x(01)00069-5. Bioorg Med Chem Lett. 2001. PMID: 11277527

2

Synthesis and histamine H3 receptor activity of 4-(n-alkyl)-1H-imidazoles and 4-(omega-phenylalkyl)-1H-imidazoles.

De Esch IJ, Gaffar A, Menge WM, Timmerman H. De Esch IJ, et al. Among authors: menge wm. Bioorg Med Chem. 1999 Dec;7(12):3003-9. doi: 10.1016/s0968-0896(99)00253-9. Bioorg Med Chem. 1999. PMID: 10658607

3

Isoquinoline and quinazoline urea analogues as antagonists for the human adenosine A(3) receptor.

van Muijlwijk-Koezen JE, Timmerman H, van der Goot H, Menge WM, Frijtag Von Drabbe Künzel J, de Groote M, IJzerman AP. van Muijlwijk-Koezen JE, et al. Among authors: menge wm. J Med Chem. 2000 Jun 1;43(11):2227-38. doi: 10.1021/jm000002u. J Med Chem. 2000. PMID: 10841801 Free article.

4

Solid-phase synthesis of 4-substituted imidazoles using a scaffold approach.

Gelens E, Koot WJ, Menge WM, Ottenheijm HC, Timmerman H. Gelens E, et al. Among authors: menge wm. Bioorg Med Chem Lett. 2000 Sep 4;10(17):1935-8. doi: 10.1016/s0960-894x(00)00363-2. Bioorg Med Chem Lett. 2000. PMID: 10987421

5

Synthesis and structure-activity relationships of conformationally constrained histamine H(3) receptor agonists.

Kitbunnadaj R, Zuiderveld OP, De Esch IJ, Vollinga RC, Bakker R, Lutz M, Spek AL, Cavoy E, Deltent MF, Menge WM, Timmerman H, Leurs R. Kitbunnadaj R, et al. Among authors: menge wm. J Med Chem. 2003 Dec 4;46(25):5445-57. doi: 10.1021/jm030905y. J Med Chem. 2003. PMID: 14640553

6

New analogs of burimamide as potent and selective histamine H3 receptor antagonists: the effect of chain length variation of the alkyl spacer and modifications of the N-thiourea substituent.

Vollinga RC, Menge WM, Leurs R, Timmerman H. Vollinga RC, et al. Among authors: menge wm. J Med Chem. 1995 Jun 9;38(12):2244-50. doi: 10.1021/jm00012a025. J Med Chem. 1995. PMID: 7783156

7

Homologs of histamine as histamine H3 receptor antagonists: a new potent and selective H3 antagonist, 4(5)-(5-aminopentyl)-1H-imidazole.

Vollinga RC, Menge WM, Leurs R, Timmerman H. Vollinga RC, et al. Among authors: menge wm. J Med Chem. 1995 Jan 20;38(2):266-71. doi: 10.1021/jm00002a008. J Med Chem. 1995. PMID: 7830269

8

A new potent and selective histamine H3 receptor agonist, 4-(1H-imidazol-4-ylmethyl)piperidine.

Vollinga RC, de Koning JP, Jansen FP, Leurs R, Menge WM, Timmerman H. Vollinga RC, et al. Among authors: menge wm. J Med Chem. 1994 Feb 4;37(3):332-3. doi: 10.1021/jm00029a002. J Med Chem. 1994. PMID: 8308858 No abstract available.

9

Characterization of the binding site of the histamine H3 receptor. 1. Various approaches to the synthesis of 2-(1H-imidazol-4-yl)cyclopropylamine and histaminergic activity of (1R,2R)- and (1S,2S)-2-(1H-imidazol-4-yl)-cyclopropylamine.

De Esch IJ, Vollinga RC, Goubitz K, Schenk H, Appelberg U, Hacksell U, Lemstra S, Zuiderveld OP, Hoffmann M, Leurs R, Menge WM, Timmerman H. De Esch IJ, et al. Among authors: menge wm. J Med Chem. 1999 Apr 8;42(7):1115-22. doi: 10.1021/jm9810912. J Med Chem. 1999. PMID: 10197956 Free article.

10

Evaluation of [18F]VUF 5000 as a potential PET ligand for brain imaging of the histamine H3 receptor.

Windhorst AD, Timmerman H, Klok RP, Menge WM, Leurs R, Herscheid JD. Windhorst AD, et al. Among authors: menge wm. Bioorg Med Chem. 1999 Sep;7(9):1761-7. doi: 10.1016/s0968-0896(99)00108-x. Bioorg Med Chem. 1999. PMID: 10530922

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