Cappelli A - Search Results

1

Mapping and fitting the peripheral benzodiazepine receptor binding site by carboxamide derivatives. Comparison of different approaches to quantitative ligand-receptor interaction modeling.

Anzini M, Cappelli A, Vomero S, Seeber M, Menziani MC, Langer T, Hagen B, Manzoni C, Bourguignon JJ. Anzini M, et al. Among authors: cappelli a. J Med Chem. 2001 Apr 12;44(8):1134-50. doi: 10.1021/jm0009742. J Med Chem. 2001. PMID: 11312914

The most potent compound, among the newly synthesized ones, shows a nanomolar PBR affinity similar to that shown by 1 and the presence of a basic N-ethyl-N-benzylaminomethyl group in 3-position of the quinoline nucleus. ...The ligand-receptor complexes obtained prov …

The most potent compound, among the newly synthesized ones, shows a nanomolar PBR affinity similar to that shown by 1 and the presenc …

2

Synthesis and benzodiazepine receptors affinity of 2,3-dihydro-9-phenyl-1H-pyrrolo[3,4-b]quinolin-1-one and 3-carbethoxy-4-phenylquinoline derivatives.

Anzini M, Cappelli A, Vomero S, Cagnotto A, Skorupska M. Anzini M, et al. Among authors: cappelli a. Farmaco. 1992 Feb;47(2):191-202. Farmaco. 1992. PMID: 1324688

3

Synthesis and 5-HT receptors binding studies of some 3-substituted-2-(4-methyl-1-piperazinyl)-4-phenylquinolines.

Anzini M, Cappelli A, Vomero S, Campiani G, Cagnotto A, Skorupska M. Anzini M, et al. Among authors: cappelli a. Farmaco. 1991 Dec;46(12):1435-47. Farmaco. 1991. PMID: 1668253

4

5-HT and benzodiazepine receptor ligands. III. Synthesis and receptor affinities of 1,2,4-triazolo[4',3':1,6]pyridazino[4,5-b]quinoline and 2,3-dihydro-9-phenyl-1H-pyrrolo[3,4-b]quinoline-1-one derivatives.

Anzini M, Cappelli A, Vomero S, Botta M, Cagnotto A. Anzini M, et al. Among authors: cappelli a. Farmaco. 1990 Nov;45(11):1169-79. Farmaco. 1990. PMID: 1965122

5

Synthesis and 5HT-receptors affinity of some 4-phenylquinoline derivatives.

Anzini M, Vomero S, Garofalo A, Cappelli A, Cagnotto A. Anzini M, et al. Among authors: cappelli a. Farmaco. 1989 Jun;44(6):555-63. Farmaco. 1989. PMID: 2529861

6

Novel, potent, and selective 5-HT3 receptor antagonists based on the arylpiperazine skeleton: synthesis, structure, biological activity, and comparative molecular field analysis studies.

Anzini M, Cappelli A, Vomero S, Giorgi G, Langer T, Hamon M, Merahi N, Emerit BM, Cagnotto A, Skorupska M, et al. Anzini M, et al. Among authors: cappelli a. J Med Chem. 1995 Jul 7;38(14):2692-704. doi: 10.1021/jm00014a021. J Med Chem. 1995. PMID: 7629808

7

Synthesis and receptor binding studies of 2-functionalized 1,4-benzodiazepine derivatives as potential metaclazepam-like antianxiety agents.

Anzini M, Cappelli A, Vomero S, Cagnotto A, Skorupska M. Anzini M, et al. Among authors: cappelli a. Farmaco. 1993 Jul;48(7):897-905. Farmaco. 1993. PMID: 8104405

8

Synthesis, biological evaluation, and quantitative receptor docking simulations of 2-[(acylamino)ethyl]-1,4-benzodiazepines as novel tifluadom-like ligands with high affinity and selectivity for kappa-opioid receptors.

Cappelli A, Anzini M, Vomero S, Menziani MC, De Benedetti PG, Sbacchi M, Clarke GD, Mennuni L. Cappelli A, et al. J Med Chem. 1996 Feb 16;39(4):860-72. doi: 10.1021/jm950423p. J Med Chem. 1996. PMID: 8632410

9

Molecular basis of peripheral vs central benzodiazepine receptor selectivity in a new class of peripheral benzodiazepine receptor ligands related to alpidem.

Anzini M, Cappelli A, Vomero S, Giorgi G, Langer T, Bruni G, Romeo MR, Basile AS. Anzini M, et al. Among authors: cappelli a. J Med Chem. 1996 Oct 11;39(21):4275-84. doi: 10.1021/jm960325j. J Med Chem. 1996. PMID: 8863805

10

Molecular structure and dynamics of some potent 5-HT3 receptor antagonists. Insight into the interaction with the receptor.

Cappelli A, Donati A, Anzini M, Vomero S, De Benedetti PG, Menziani MC, Langer T. Cappelli A, et al. Bioorg Med Chem. 1996 Aug;4(8):1255-69. doi: 10.1016/0968-0896(96)00122-8. Bioorg Med Chem. 1996. PMID: 8879547

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