Sakashita H - Search Results

1

Synthesis, structure-activity relationships, and pharmacokinetic profiles of nonpeptidic alpha-keto heterocycles as novel inhibitors of human chymase.

Akahoshi F, Ashimori A, Sakashita H, Yoshimura T, Imada T, Nakajima M, Mitsutomi N, Kuwahara S, Ohtsuka T, Fukaya C, Miyazaki M, Nakamura N. Akahoshi F, et al. Among authors: sakashita h. J Med Chem. 2001 Apr 12;44(8):1286-96. doi: 10.1021/jm000496v. J Med Chem. 2001. PMID: 11312927

2

Syntheses and evaluation of amidinobenzofuran derivatives as tryptase inhibitors.

Ono S, Kuwahara S, Takeuchi M, Sakashita H, Naito Y, Kondo T. Ono S, et al. Among authors: sakashita h. Bioorg Med Chem Lett. 1999 Dec 6;9(23):3285-90. doi: 10.1016/s0960-894x(99)00594-6. Bioorg Med Chem Lett. 1999. PMID: 10612586

3

Synthesis, structure-activity relationships, and pharmacokinetic profiles of nonpeptidic difluoromethylene ketones as novel inhibitors of human chymase.

Akahoshi F, Ashimori A, Sakashita H, Yoshimura T, Eda M, Imada T, Nakajima M, Mitsutomi N, Kuwahara S, Ohtsuka T, Fukaya C, Miyazaki M, Nakamura N. Akahoshi F, et al. Among authors: sakashita h. J Med Chem. 2001 Apr 12;44(8):1297-304. doi: 10.1021/jm000497n. J Med Chem. 2001. PMID: 11312928

4

Novel potassium channel openers: synthesis and pharmacological evaluation of new N-(substituted-3-pyridyl)-N'-alkylthioureas and related compounds.

Takemoto T, Eda M, Okada T, Sakashita H, Matzno S, Gohda M, Ebisu H, Nakamura N, Fukaya C, Hihara M, et al. Takemoto T, et al. Among authors: sakashita h. J Med Chem. 1994 Jan 7;37(1):18-25. doi: 10.1021/jm00027a003. J Med Chem. 1994. PMID: 8289193

5

Synthesis and pharmacological evaluation of N-(6-functionalized-amino-3-pyridyl)-N'-bicycloalkyl-N''-cyanoguanidine s as antihypertensive agents.

Eda M, Takemoto T, Okada T, Sakashita H, Matzno S, Gohda M, Hayashi K, Nakamura N, Fukaya C. Eda M, et al. Among authors: sakashita h. Chem Pharm Bull (Tokyo). 1996 Feb;44(2):307-13. doi: 10.1248/cpb.44.307. Chem Pharm Bull (Tokyo). 1996. PMID: 8998837

6

Novel histamine H3 receptor antagonists: synthesis and evaluation of formamidine and S-methylisothiourea derivatives.

Goto T, Sakashita H, Murakami K, Sugiura M, Kondo T, Fukaya C. Goto T, et al. Among authors: sakashita h. Chem Pharm Bull (Tokyo). 1997 Feb;45(2):305-11. doi: 10.1248/cpb.45.305. Chem Pharm Bull (Tokyo). 1997. PMID: 9118445

7

Coumarin and chromen-4-one analogues as tautomerase inhibitors of macrophage migration inhibitory factor: discovery and X-ray crystallography.

Orita M, Yamamoto S, Katayama N, Aoki M, Takayama K, Yamagiwa Y, Seki N, Suzuki H, Kurihara H, Sakashita H, Takeuchi M, Fujita S, Yamada T, Tanaka A. Orita M, et al. Among authors: sakashita h. J Med Chem. 2001 Feb 15;44(4):540-7. doi: 10.1021/jm000386o. J Med Chem. 2001. PMID: 11170644

8

Real-time measurements of spatial velocity distribution with a laser Doppler imaging system.

Yoshimura T, Sakashita H, Wakabayashi N. Yoshimura T, et al. Among authors: sakashita h. Appl Opt. 1983 Aug 15;22(16):2448-52. doi: 10.1364/ao.22.002448. Appl Opt. 1983. PMID: 18196154

9

4-Hydroxypyridazin-3(2H)-one derivatives as novel D-amino acid oxidase inhibitors.

Hondo T, Warizaya M, Niimi T, Namatame I, Yamaguchi T, Nakanishi K, Hamajima T, Harada K, Sakashita H, Matsumoto Y, Orita M, Takeuchi M. Hondo T, et al. Among authors: sakashita h. J Med Chem. 2013 May 9;56(9):3582-92. doi: 10.1021/jm400095b. Epub 2013 Apr 25. J Med Chem. 2013. PMID: 23566269

10

Design and synthesis of non-peptidic inhibitors for the Syk C-terminal SH2 domain based on structure-based in-silico screening.

Niimi T, Orita M, Okazawa-Igarashi M, Sakashita H, Kikuchi K, Ball E, Ichikawa A, Yamagiwa Y, Sakamoto S, Tanaka A, Tsukamoto S, Fujita S, Tatsuta K, Maeda Y, Chikauchi K. Niimi T, et al. Among authors: sakashita h. J Med Chem. 2001 Dec 20;44(26):4737-40. doi: 10.1021/jm010313k. J Med Chem. 2001. PMID: 11741491

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

241 results

Search Page

Filters