Brun R - Search Results

1

Novel inhibitors of Leishmanial dihydrofolate reductase.

Chowdhury SF, Di Lucrezia R, Guerrero RH, Brun R, Goodman J, Ruiz-Perez LM, Pacanowska DG, Gilbert IH. Chowdhury SF, et al. Among authors: brun r. Bioorg Med Chem Lett. 2001 Apr 23;11(8):977-80. doi: 10.1016/s0960-894x(01)00089-0. Bioorg Med Chem Lett. 2001. PMID: 11327604

2

Design, synthesis and evaluation of novel uracil amino acid conjugates for the inhibition of Trypanosoma cruzi dUTPase.

Mc Carthy OK, Schipani A, Buendía AM, Ruiz-Perez LM, Kaiser M, Brun R, Pacanowska DG, Gilbert IH. Mc Carthy OK, et al. Among authors: brun r. Bioorg Med Chem Lett. 2006 Jul 15;16(14):3809-12. doi: 10.1016/j.bmcl.2006.04.027. Epub 2006 May 3. Bioorg Med Chem Lett. 2006. PMID: 16677813

3

Acyclic nucleoside analogues as inhibitors of Plasmodium falciparum dUTPase.

Nguyen C, Ruda GF, Schipani A, Kasinathan G, Leal I, Musso-Buendia A, Kaiser M, Brun R, Ruiz-Pérez LM, Sahlberg BL, Johansson NG, Gonzalez-Pacanowska D, Gilbert IH. Nguyen C, et al. Among authors: brun r. J Med Chem. 2006 Jul 13;49(14):4183-95. doi: 10.1021/jm060126s. J Med Chem. 2006. PMID: 16821778

4

Design, synthesis and evaluation of novel uracil acetamide derivatives as potential inhibitors of Plasmodium falciparum dUTP nucleotidohydrolase.

McCarthy O, Musso-Buendia A, Kaiser M, Brun R, Ruiz-Perez LM, Johansson NG, Pacanowska DG, Gilbert IH. McCarthy O, et al. Among authors: brun r. Eur J Med Chem. 2009 Feb;44(2):678-88. doi: 10.1016/j.ejmech.2008.05.018. Epub 2008 Jul 10. Eur J Med Chem. 2009. PMID: 18619713

5

Selective inhibition of Trypanosoma brucei 6-phosphogluconate dehydrogenase by high-energy intermediate and transition-state analogues.

Dardonville C, Rinaldi E, Barrett MP, Brun R, Gilbert IH, Hanau S. Dardonville C, et al. Among authors: brun r. J Med Chem. 2004 Jun 17;47(13):3427-37. doi: 10.1021/jm031066i. J Med Chem. 2004. PMID: 15189039

6

Design, synthesis and evaluation of 2,4-diaminoquinazolines as inhibitors of trypanosomal and leishmanial dihydrofolate reductase.

Khabnadideh S, Pez D, Musso A, Brun R, Pérez LM, González-Pacanowska D, Gilbert IH. Khabnadideh S, et al. Among authors: brun r. Bioorg Med Chem. 2005 Apr 1;13(7):2637-49. doi: 10.1016/j.bmc.2005.01.025. Bioorg Med Chem. 2005. PMID: 15755663

7

Design and synthesis of a series of melamine-based nitroheterocycles with activity against Trypanosomatid parasites.

Baliani A, Bueno GJ, Stewart ML, Yardley V, Brun R, Barrett MP, Gilbert IH. Baliani A, et al. Among authors: brun r. J Med Chem. 2005 Aug 25;48(17):5570-9. doi: 10.1021/jm050177+. J Med Chem. 2005. PMID: 16107157

8

Deoxyuridine triphosphate nucleotidohydrolase as a potential antiparasitic drug target.

Nguyen C, Kasinathan G, Leal-Cortijo I, Musso-Buendia A, Kaiser M, Brun R, Ruiz-Pérez LM, Johansson NG, González-Pacanowska D, Gilbert IH. Nguyen C, et al. Among authors: brun r. J Med Chem. 2005 Sep 22;48(19):5942-54. doi: 10.1021/jm050111e. J Med Chem. 2005. PMID: 16161998

9

Synthesis and testing of 5-benzyl-2,4-diaminopyrimidines as potential inhibitors of leishmanial and trypanosomal dihydrofolate reductase.

Chowdhury SF, Guerrero RH, Brun R, Ruiz-Perez LM, Pacanowska DG, Gilbert IH. Chowdhury SF, et al. Among authors: brun r. J Enzyme Inhib Med Chem. 2002 Oct;17(5):293-302. doi: 10.1080/1475636021000059083. J Enzyme Inhib Med Chem. 2002. PMID: 12683746

10

Synthesis and biological evaluation of substrate-based inhibitors of 6-phosphogluconate dehydrogenase as potential drugs against African trypanosomiasis.

Dardonville C, Rinaldi E, Hanau S, Barrett MP, Brun R, Gilbert IH. Dardonville C, et al. Among authors: brun r. Bioorg Med Chem. 2003 Jul 17;11(14):3205-14. doi: 10.1016/s0968-0896(03)00191-3. Bioorg Med Chem. 2003. PMID: 12818683

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