Masciadri R - Search Results

1

2-(2-Oxo-1,4-dihydro-2H-quinazolin-3-yl)- and 2-(2,2-dioxo-1,4-dihydro-2H-2lambda6-benzo[1,2,6]thiadiazin-3-yl)-N-hydroxy-acetamides as potent and selective peptide deformylase inhibitors.

Apfel C, Banner DW, Bur D, Dietz M, Hubschwerlen C, Locher H, Marlin F, Masciadri R, Pirson W, Stalder H. Apfel C, et al. Among authors: masciadri r. J Med Chem. 2001 Jun 7;44(12):1847-52. doi: 10.1021/jm000352g. J Med Chem. 2001. PMID: 11384231

2

New antibacterial agents derived from the DNA gyrase inhibitor cyclothialidine.

Angehrn P, Buchmann S, Funk C, Goetschi E, Gmuender H, Hebeisen P, Kostrewa D, Link H, Luebbers T, Masciadri R, Nielsen J, Reindl P, Ricklin F, Schmitt-Hoffmann A, Theil FP. Angehrn P, et al. Among authors: masciadri r. J Med Chem. 2004 Mar 11;47(6):1487-513. doi: 10.1021/jm0310232. J Med Chem. 2004. PMID: 14998336

3

Discovery of tetrahydro-cyclopenta[b]indole as selective LXRs modulator.

Ratni H, Blum-Kaelin D, Dehmlow H, Hartman P, Jablonski P, Masciadri R, Maugeais C, Patiny-Adam A, Panday N, Wright M. Ratni H, et al. Among authors: masciadri r. Bioorg Med Chem Lett. 2009 Mar 15;19(6):1654-7. doi: 10.1016/j.bmcl.2009.01.109. Epub 2009 Feb 6. Bioorg Med Chem Lett. 2009. PMID: 19231176

4

Discovery of the imidazo[1,5-a][1,2,4]-triazolo[1,5-d][1,4]benzodiazepine scaffold as a novel, potent and selective GABA(A) alpha5 inverse agonist series.

Achermann G, Ballard TM, Blasco F, Broutin PE, Büttelmann B, Fischer H, Graf M, Hernandez MC, Hilty P, Knoflach F, Koblet A, Knust H, Kurt A, Martin JR, Masciadri R, Porter RH, Stadler H, Thomas AW, Trube G, Wichmann J. Achermann G, et al. Among authors: masciadri r. Bioorg Med Chem Lett. 2009 Oct 1;19(19):5746-52. doi: 10.1016/j.bmcl.2009.07.153. Epub 2009 Aug 4. Bioorg Med Chem Lett. 2009. PMID: 19726184

5

Cyclothialidine and its congeners: a new class of DNA gyrase inhibitors.

Goetschi E, Angehrn P, Gmuender H, Hebeisen P, Link H, Masciadri R, Nielsen J. Goetschi E, et al. Among authors: masciadri r. Pharmacol Ther. 1993 Nov;60(2):367-80. doi: 10.1016/0163-7258(93)90017-8. Pharmacol Ther. 1993. PMID: 8022866 Review.

6

Efficient Fluorination with Tetrabutylammonium Dihydrogen Trifluoride in a Novel Approach toward 1-alpha-Fluoro-25-hydroxy-vitamin D(3) Analogues.

Barbier P, Mohr P, Muller M, Masciadri R. Barbier P, et al. Among authors: masciadri r. J Org Chem. 1998 Oct 2;63(20):6984-6989. doi: 10.1021/jo980764l. J Org Chem. 1998. PMID: 11672321

7

Ro 42-1611 (arteflene), a new effective antimalarial: chemical structure and biological activity.

Hofheinz W, Bürgin H, Gocke E, Jaquet C, Masciadri R, Schmid G, Stohler H, Urwyler H. Hofheinz W, et al. Among authors: masciadri r. Trop Med Parasitol. 1994 Sep;45(3):261-5. Trop Med Parasitol. 1994. PMID: 7899801

8

Antimalarial activity of the bisquinoline trans-N1,N2-bis (7-chloroquinolin-4-yl)cyclohexane-1,2-diamine: comparison of two stereoisomers and detailed evaluation of the S,S enantiomer, Ro 47-7737.

Ridley RG, Matile H, Jaquet C, Dorn A, Hofheinz W, Leupin W, Masciadri R, Theil FP, Richter WF, Girometta MA, Guenzi A, Urwyler H, Gocke E, Potthast JM, Csato M, Thomas A, Peters W. Ridley RG, et al. Among authors: masciadri r. Antimicrob Agents Chemother. 1997 Mar;41(3):677-86. doi: 10.1128/AAC.41.3.677. Antimicrob Agents Chemother. 1997. PMID: 9056013 Free PMC article.

9

Characterization of (R,S)-5,7-di-tert-butyl-3-hydroxy-3-trifluoromethyl-3H-benzofuran-2-one as a positive allosteric modulator of GABAB receptors.

Malherbe P, Masciadri R, Norcross RD, Knoflach F, Kratzeisen C, Zenner MT, Kolb Y, Marcuz A, Huwyler J, Nakagawa T, Porter RH, Thomas AW, Wettstein JG, Sleight AJ, Spooren W, Prinssen EP. Malherbe P, et al. Among authors: masciadri r. Br J Pharmacol. 2008 Jun;154(4):797-811. doi: 10.1038/bjp.2008.135. Epub 2008 Apr 21. Br J Pharmacol. 2008. PMID: 18536733 Free PMC article.

10

4-aminoquinoline analogs of chloroquine with shortened side chains retain activity against chloroquine-resistant Plasmodium falciparum.

Ridley RG, Hofheinz W, Matile H, Jaquet C, Dorn A, Masciadri R, Jolidon S, Richter WF, Guenzi A, Girometta MA, Urwyler H, Huber W, Thaithong S, Peters W. Ridley RG, et al. Among authors: masciadri r. Antimicrob Agents Chemother. 1996 Aug;40(8):1846-54. doi: 10.1128/AAC.40.8.1846. Antimicrob Agents Chemother. 1996. PMID: 8843292 Free PMC article.

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