Trincavelli L - Search Results

1

Novel N-(arylalkyl)indol-3-ylglyoxylylamides targeted as ligands of the benzodiazepine receptor: synthesis, biological evaluation, and molecular modeling analysis of the structure-activity relationships.

Primofiore G, Settimo FD, Taliani S, Marini AM, Novellino E, Greco G, Lavecchia A, Besnard F, Trincavelli L, Costa B, Martini C. Primofiore G, et al. Among authors: trincavelli l. J Med Chem. 2001 Jul 5;44(14):2286-97. doi: 10.1021/jm010827j. J Med Chem. 2001. PMID: 11428922

2

Design, synthesis and biological evaluation of novel N-alkyl- and N-acyl-(7-substituted-2-phenylimidazo[1,2-a][1,3,5]triazin-4-yl)amines (ITAs) as novel A(1) adenosine receptor antagonists.

Novellino E, Abignente E, Cosimelli B, Greco G, Iadanza M, Laneri S, Lavecchia A, Rimoli MG, Settimo FD, Primofiore G, Tuscano D, Trincavelli L, Martini C. Novellino E, et al. Among authors: trincavelli l. J Med Chem. 2002 Nov 7;45(23):5030-6. doi: 10.1021/jm020911e. J Med Chem. 2002. PMID: 12408713

3

Geometrically constrained analogues of N-benzylindolylglyoxylylamides: [1, 2, 4]triazino[4, 3-a]benzimidazol-4(10H)-one derivatives as potential new ligands at the benzodiazepine receptor.

Primofiore G, Da Settimo F, Taliani S, Marini AM, Simorini F, Novellino E, Greco G, Trincavelli L, Martini C. Primofiore G, et al. Among authors: trincavelli l. Arch Pharm (Weinheim). 2003 Sep;336(9):413-21. doi: 10.1002/ardp.200300788. Arch Pharm (Weinheim). 2003. PMID: 14528489

4

Synthesis and benzodiazepine receptor affinity of derivatives of the new tricyclic heteroaromatic system pyrido[3',2':5,6]thiopyrano[4,3-c]pyridazin-3(2H,5H)-one.

Primofiore G, Da Settimo F, Marini AM, Simorini F, La Motta C, Taliani S, Laneri S, Trincavelli L, Martini C. Primofiore G, et al. Among authors: trincavelli l. Arch Pharm (Weinheim). 2005 Mar;338(2-3):126-32. doi: 10.1002/ardp.200400948. Arch Pharm (Weinheim). 2005. PMID: 15799013

5

Isosteric replacement of amide by ester function. Synthesis and benzodiazepine receptor affinity of indol-3-ylglyoxylyl ester derivatives.

Da Settimo A, Primofiore G, Marini AM, Da Settimo F, Nuti V, Martini C, Trincavelli L, Lucacchini A. Da Settimo A, et al. Among authors: trincavelli l. Farmaco. 1997 Jun-Jul;52(6-7):421-8. Farmaco. 1997. PMID: 9372593

6

3-Aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: tricyclic heteroaromatic derivatives as a new class of benzodiazepine receptor ligands.

Primofiore G, Da Settimo F, Taliani S, Marini AM, La Motta C, Novellino E, Greco G, Gesi M, Trincavelli L, Martini C. Primofiore G, et al. Among authors: trincavelli l. J Med Chem. 2000 Jan 13;43(1):96-102. doi: 10.1021/jm991131h. J Med Chem. 2000. PMID: 10633040

7

1,2,4-Triazolo[4,3-a]quinoxalin-1-one: a versatile tool for the synthesis of potent and selective adenosine receptor antagonists.

Colotta V, Catarzi D, Varano F, Cecchi L, Filacchioni G, Martini C, Trincavelli L, Lucacchini A. Colotta V, et al. Among authors: trincavelli l. J Med Chem. 2000 Mar 23;43(6):1158-64. doi: 10.1021/jm991096e. J Med Chem. 2000. PMID: 10737748

8

Synthesis and structure-activity relationships of a new set of 2-arylpyrazolo[3,4-c]quinoline derivatives as adenosine receptor antagonists.

Colotta V, Catarzi D, Varano F, Cecchi L, Filacchioni G, Martini C, Trincavelli L, Lucacchini A. Colotta V, et al. Among authors: trincavelli l. J Med Chem. 2000 Aug 10;43(16):3118-24. doi: 10.1021/jm000936i. J Med Chem. 2000. PMID: 10956220

9

3-Aryl[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: a new class of selective A1 adenosine receptor antagonists.

Da Settimo F, Primofiore G, Taliani S, Marini AM, La Motta C, Novellino E, Greco G, Lavecchia A, Trincavelli L, Martini C. Da Settimo F, et al. Among authors: trincavelli l. J Med Chem. 2001 Feb 1;44(3):316-27. doi: 10.1021/jm001054m. J Med Chem. 2001. PMID: 11462973

10

Synthesis and structure-activity relationships of a new set of 1,2,4-triazolo[4,3-a]quinoxalin-1-one derivatives as adenosine receptor antagonists.

Colotta V, Catarzi D, Varano F, Filacchioni G, Martini C, Trincavelli L, Lucacchini A. Colotta V, et al. Among authors: trincavelli l. Bioorg Med Chem. 2003 Aug 5;11(16):3541-50. doi: 10.1016/s0968-0896(03)00338-9. Bioorg Med Chem. 2003. PMID: 12878146

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