Grellepois F - Search Results

1

Anhydrodihydroartemisinin and its 10-trifluoromethyl analogue: access to novel d-ring-contracted artemisinin trifluoromethyl ketones.

Grellepois F, Chorki F, Crousse B, Ourévitch M, Bonnet-Delpon D, Bégué JP. Grellepois F, et al. J Org Chem. 2002 Feb 22;67(4):1253-60. doi: 10.1021/jo016091f. J Org Chem. 2002. PMID: 11846670

2

First synthesis of 10 alpha-(trifluoromethyl)deoxoartemisinin.

Chorki F, Grellepois F, Crousse B, Hoang VD, Hung NV, Bonnet-Delpon D, Bégué JP. Chorki F, et al. Among authors: grellepois f. Org Lett. 2002 Mar 7;4(5):757-9. doi: 10.1021/ol017227z. Org Lett. 2002. PMID: 11869120

3

Orally active antimalarials: hydrolytically stable derivatives of 10-trifluoromethyl anhydrodihydroartemisinin.

Grellepois F, Chorki F, Ourévitch M, Charneau S, Grellier P, McIntosh KA, Charman WN, Pradines B, Crousse B, Bonnet-Delpon D, Bégué JP. Grellepois F, et al. J Med Chem. 2004 Mar 11;47(6):1423-33. doi: 10.1021/jm030947m. J Med Chem. 2004. PMID: 14998331

4

Synthesis of new artemisinin-derived dimers by self-cross-metathesis reaction.

Grellepois F, Crousse B, Bonnet-Delpon D, Bégué JP. Grellepois F, et al. Org Lett. 2005 Nov 10;7(23):5219-22. doi: 10.1021/ol052056+. Org Lett. 2005. PMID: 16268542

5

Fluoro artemisinins: difluoromethylene ketones.

Chorki F, Grellepois F, Crousse B, Ourévitch M, Bonnet-Delpon D, Bégué JP. Chorki F, et al. Among authors: grellepois f. J Org Chem. 2001 Nov 16;66(23):7858-63. doi: 10.1021/jo0158579. J Org Chem. 2001. PMID: 11701047

6

Design, synthesis and antimalarial activity of trifluoromethylartemisinin-mefloquine dual molecules.

Grellepois F, Grellier P, Bonnet-Delpon D, Bégué JP. Grellepois F, et al. Chembiochem. 2005 Apr;6(4):648-52. doi: 10.1002/cbic.200400347. Chembiochem. 2005. PMID: 15723441 No abstract available.

7

Enantiopure quaternary alpha-trifluoromethyl-alpha-alkoxyaldehydes from L-tartaric acid derived ketoamides.

Nonnenmacher J, Massicot F, Grellepois F, Portella C. Nonnenmacher J, et al. Among authors: grellepois f. J Org Chem. 2008 Oct 17;73(20):7990-5. doi: 10.1021/jo8013403. Epub 2008 Sep 25. J Org Chem. 2008. PMID: 18816141

8

Enantiopure trifluoromethylated β(3,3)-amino acids: synthesis by asymmetric Reformatsky reaction with stable analogues of trifluoromethyl N-tert-butanesulfinylketoimines and incorporation into α/β-peptides.

Grellepois F. Grellepois F. J Org Chem. 2013 Feb 1;78(3):1127-37. doi: 10.1021/jo302549v. Epub 2013 Jan 8. J Org Chem. 2013. PMID: 23273379

9

Enantiomerically pure 2-aryl(alkyl)-2-trifluoromethylaziridines: synthesis and ring opening with selected O- and N-nucleophiles.

Grellepois F, Nonnenmacher J, Lachaud F, Portella C. Grellepois F, et al. Org Biomol Chem. 2011 Feb 21;9(4):1160-8. doi: 10.1039/c0ob00690d. Epub 2010 Dec 15. Org Biomol Chem. 2011. PMID: 21157614

10

cis-Dihydroxylated α-Trifluoromethylated N,O-Acetal from l-Tartaric Acid: Synthesis of Tetrasubstituted Stereocenter via Diastereoselective Pictet-Spengler Cyclization of N-Acyliminium Ions.

Ben Jamaa A, Latrache M, Riguet E, Grellepois F. Ben Jamaa A, et al. Among authors: grellepois f. J Org Chem. 2020 Aug 7;85(15):9585-9598. doi: 10.1021/acs.joc.0c00801. Epub 2020 Jul 26. J Org Chem. 2020. PMID: 32790358

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