Boivin RP - Search Results

1

A concerted, rational design of type 1 17beta-hydroxysteroid dehydrogenase inhibitors: estradiol-adenosine hybrids with high affinity.

Qiu W, Campbell RL, Gangloff A, Dupuis P, Boivin RP, Tremblay MR, Poirier D, Lin SX. Qiu W, et al. Among authors: boivin rp. FASEB J. 2002 Nov;16(13):1829-31. doi: 10.1096/fj.02-0026fje. Epub 2002 Sep 5. FASEB J. 2002. PMID: 12223444

2

Inhibitors of type 1 17beta-hydroxysteroid dehydrogenase with reduced estrogenic activity: modifications of the positions 3 and 6 of estradiol.

Tremblay MR, Boivin RP, Luu-The V, Poirier D. Tremblay MR, et al. Among authors: boivin rp. J Enzyme Inhib Med Chem. 2005 Apr;20(2):153-63. doi: 10.1080/14756360500043307. J Enzyme Inhib Med Chem. 2005. PMID: 15968820 Free article.

3

Estrone and estradiol C-16 derivatives as inhibitors of type 1 17beta-hydroxysteroid dehydrogenase.

Poirier D, Chang HJ, Azzi A, Boivin RP, Lin SX. Poirier D, et al. Among authors: boivin rp. Mol Cell Endocrinol. 2006 Mar 27;248(1-2):236-8. doi: 10.1016/j.mce.2005.10.017. Epub 2005 Dec 7. Mol Cell Endocrinol. 2006. PMID: 16337735

4

Estradiol-adenosine hybrid compounds designed to inhibit type 1 17beta-hydroxysteroid dehydrogenase.

Poirier D, Boivin RP, Tremblay MR, Bérubé M, Qiu W, Lin SX. Poirier D, et al. Among authors: boivin rp. J Med Chem. 2005 Dec 29;48(26):8134-47. doi: 10.1021/jm058235e. J Med Chem. 2005. PMID: 16366595

5

C16 and C17 derivatives of estradiol as inhibitors of 17 beta-hydroxysteroid dehydrogenase type 1: chemical synthesis and structure-activity relationships.

Sam KM, Boivin RP, Tremblay MR, Auger S, Poirier D. Sam KM, et al. Among authors: boivin rp. Drug Des Discov. 1998 May;15(3):157-80. Drug Des Discov. 1998. PMID: 9689499

6

3Beta-sulfamate derivatives of C19 and C21 steroids bearing a t-butylbenzyl or a benzyl group: synthesis and evaluation as non-estrogenic and non-androgenic steroid sulfatase inhibitors.

Ciobanu LC, Boivin RP, Luu-The V, Poirier D. Ciobanu LC, et al. Among authors: boivin rp. J Enzyme Inhib Med Chem. 2003 Feb;18(1):15-26. doi: 10.1080/1475636031000069282. J Enzyme Inhib Med Chem. 2003. PMID: 12751816 Free article.

7

17 alpha-alkyl- or 17 alpha-substituted benzyl-17 beta-estradiols: a new family of estrone-sulfatase inhibitors.

Poirier D, Boivin RP. Poirier D, et al. Among authors: boivin rp. Bioorg Med Chem Lett. 1998 Jul 21;8(14):1891-6. doi: 10.1016/s0960-894x(98)00330-8. Bioorg Med Chem Lett. 1998. PMID: 9873454

8

17Alpha-alkan (or alkyn) amide derivatives of estradiol as inhibitors of steroid-sulfatase activity.

Boivin RP, Labrie F, Poirier D. Boivin RP, et al. Steroids. 1999 Dec;64(12):825-33. doi: 10.1016/s0039-128x(99)00060-4. Steroids. 1999. PMID: 10576217

9

Structure-activity relationships of 17alpha-derivatives of estradiol as inhibitors of steroid sulfatase.

Boivin RP, Luu-The V, Lachance R, Labrie F, Poirier D. Boivin RP, et al. J Med Chem. 2000 Nov 16;43(23):4465-78. doi: 10.1021/jm0001166. J Med Chem. 2000. PMID: 11087571

10

Potent inhibition of steroid sulfatase activity by 3-O-sulfamate 17alpha-benzyl(or 4'-tert-butylbenzyl)estra-1,3,5(10)-trienes: combination of two substituents at positions C3 and c17alpha of estradiol.

Ciobanu LC, Boivin RP, Luu-The V, Labrie F, Poirier D. Ciobanu LC, et al. Among authors: boivin rp. J Med Chem. 1999 Jun 17;42(12):2280-6. doi: 10.1021/jm980677l. J Med Chem. 1999. PMID: 10377235

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