Burstein ES - Search Results

1

Discovery of the first nonpeptide agonist of the GPR14/urotensin-II receptor: 3-(4-chlorophenyl)-3-(2- (dimethylamino)ethyl)isochroman-1-one (AC-7954).

Croston GE, Olsson R, Currier EA, Burstein ES, Weiner D, Nash N, Severance D, Allenmark SG, Thunberg L, Ma JN, Mohell N, O'Dowd B, Brann MR, Hacksell U. Croston GE, et al. Among authors: burstein es. J Med Chem. 2002 Nov 7;45(23):4950-3. doi: 10.1021/jm025551+. J Med Chem. 2002. PMID: 12408704

2

Discovery of potent and selective small-molecule PAR-2 agonists.

Seitzberg JG, Knapp AE, Lund BW, Mandrup Bertozzi S, Currier EA, Ma JN, Sherbukhin V, Burstein ES, Olsson R. Seitzberg JG, et al. Among authors: burstein es. J Med Chem. 2008 Sep 25;51(18):5490-3. doi: 10.1021/jm800754r. Epub 2008 Aug 23. J Med Chem. 2008. PMID: 18720984

3

Discovery of non-peptidergic MrgX1 and MrgX2 receptor agonists and exploration of an initial SAR using solid-phase synthesis.

Malik L, Kelly NM, Ma JN, Currier EA, Burstein ES, Olsson R. Malik L, et al. Among authors: burstein es. Bioorg Med Chem Lett. 2009 Mar 15;19(6):1729-32. doi: 10.1016/j.bmcl.2009.01.085. Epub 2009 Jan 30. Bioorg Med Chem Lett. 2009. PMID: 19230660

4

Synthesis and evaluation of dibenzothiazepines: a novel class of selective cannabinoid-1 receptor inverse agonists.

Pettersson H, Bülow A, Ek F, Jensen J, Ottesen LK, Fejzic A, Ma JN, Del Tredici AL, Currier EA, Gardell LR, Tabatabaei A, Craig D, McFarland K, Ott TR, Piu F, Burstein ES, Olsson R. Pettersson H, et al. Among authors: burstein es. J Med Chem. 2009 Apr 9;52(7):1975-82. doi: 10.1021/jm801534c. J Med Chem. 2009. PMID: 19338356

5

Optimization of isochromanone based urotensin II receptor agonists.

Lehmann F, Currier EA, Olsson R, Ma JN, Burstein ES, Hacksell U, Luthman K. Lehmann F, et al. Among authors: burstein es. Bioorg Med Chem. 2010 Jul 1;18(13):4844-54. doi: 10.1016/j.bmc.2010.04.041. Epub 2010 Jun 1. Bioorg Med Chem. 2010. PMID: 20570157

6

Discovery of a class of calcium sensing receptor positive allosteric modulators; 1-(benzothiazol-2-yl)-1-phenylethanols.

Gustafsson M, Jensen J, Bertozzi SM, Currier EA, Ma JN, Burstein ES, Olsson R. Gustafsson M, et al. Among authors: burstein es. Bioorg Med Chem Lett. 2010 Oct 1;20(19):5918-21. doi: 10.1016/j.bmcl.2010.07.077. Epub 2010 Jul 23. Bioorg Med Chem Lett. 2010. PMID: 20727747

7

Discovery of an ectopic activation site on the M(1) muscarinic receptor.

Spalding TA, Trotter C, Skjaerbaek N, Messier TL, Currier EA, Burstein ES, Li D, Hacksell U, Brann MR. Spalding TA, et al. Among authors: burstein es. Mol Pharmacol. 2002 Jun;61(6):1297-302. doi: 10.1124/mol.61.6.1297. Mol Pharmacol. 2002. PMID: 12021390

8

Discovery of novel peptide/receptor interactions: identification of PHM-27 as a potent agonist of the human calcitonin receptor.

Ma JN, Currier EA, Essex A, Feddock M, Spalding TA, Nash NR, Brann MR, Burstein ES. Ma JN, et al. Among authors: burstein es. Biochem Pharmacol. 2004 Apr 1;67(7):1279-84. doi: 10.1016/j.bcp.2003.11.008. Biochem Pharmacol. 2004. PMID: 15013843

9

Pharmacology of polymorphic variants of the human 5-HT1A receptor.

Del Tredici AL, Schiffer HH, Burstein ES, Lameh J, Mohell N, Hacksell U, Brann MR, Weiner DM. Del Tredici AL, et al. Among authors: burstein es. Biochem Pharmacol. 2004 Feb 1;67(3):479-90. doi: 10.1016/j.bcp.2003.09.030. Biochem Pharmacol. 2004. PMID: 15037200

10

Characterization of the Mas-related gene family: structural and functional conservation of human and rhesus MrgX receptors.

Burstein ES, Ott TR, Feddock M, Ma JN, Fuhs S, Wong S, Schiffer HH, Brann MR, Nash NR. Burstein ES, et al. Br J Pharmacol. 2006 Jan;147(1):73-82. doi: 10.1038/sj.bjp.0706448. Br J Pharmacol. 2006. PMID: 16284629 Free PMC article.

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