Arndt K - Search Results

1

SKI-606, a 4-anilino-3-quinolinecarbonitrile dual inhibitor of Src and Abl kinases, is a potent antiproliferative agent against chronic myelogenous leukemia cells in culture and causes regression of K562 xenografts in nude mice.

Golas JM, Arndt K, Etienne C, Lucas J, Nardin D, Gibbons J, Frost P, Ye F, Boschelli DH, Boschelli F. Golas JM, et al. Among authors: arndt k. Cancer Res. 2003 Jan 15;63(2):375-81. Cancer Res. 2003. PMID: 12543790

2

SKI-606, a Src/Abl inhibitor with in vivo activity in colon tumor xenograft models.

Golas JM, Lucas J, Etienne C, Golas J, Discafani C, Sridharan L, Boghaert E, Arndt K, Ye F, Boschelli DH, Li F, Titsch C, Huselton C, Chaudhary I, Boschelli F. Golas JM, et al. Among authors: arndt k. Cancer Res. 2005 Jun 15;65(12):5358-64. doi: 10.1158/0008-5472.CAN-04-2484. Cancer Res. 2005. PMID: 15958584

3

Bosutinib: a review of preclinical studies in chronic myelogenous leukaemia.

Boschelli F, Arndt K, Gambacorti-Passerini C. Boschelli F, et al. Among authors: arndt k. Eur J Cancer. 2010 Jul;46(10):1781-9. doi: 10.1016/j.ejca.2010.02.032. Eur J Cancer. 2010. PMID: 20399641 Review.

4

Optimization of 4-phenylamino-3-quinolinecarbonitriles as potent inhibitors of Src kinase activity.

Boschelli DH, Ye F, Wang YD, Dutia M, Johnson SL, Wu B, Miller K, Powell DW, Yaczko D, Young M, Tischler M, Arndt K, Discafani C, Etienne C, Gibbons J, Grod J, Lucas J, Weber JM, Boschelli F. Boschelli DH, et al. Among authors: arndt k. J Med Chem. 2001 Nov 8;44(23):3965-77. doi: 10.1021/jm0102250. J Med Chem. 2001. PMID: 11689083

5

IkappaBalpha kinase inhibitor IKI-1 conferred tumor necrosis factor alpha sensitivity to pancreatic cancer cells and a xenograft tumor model.

Zhang Y, Gavriil M, Lucas J, Mandiyan S, Follettie M, Diesl V, Sum FW, Powell D, Haney S, Abraham R, Arndt K. Zhang Y, et al. Among authors: arndt k. Cancer Res. 2008 Nov 15;68(22):9519-24. doi: 10.1158/0008-5472.CAN-08-1549. Cancer Res. 2008. PMID: 19010928

6

Synthesis and Src kinase inhibitory activity of a series of 4-phenylamino-3-quinolinecarbonitriles.

Boschelli DH, Wang YD, Ye F, Wu B, Zhang N, Dutia M, Powell DW, Wissner A, Arndt K, Weber JM, Boschelli F. Boschelli DH, et al. Among authors: arndt k. J Med Chem. 2001 Mar 1;44(5):822-33. doi: 10.1021/jm000420z. J Med Chem. 2001. PMID: 11262092

7

A cell-based screen for inhibitors of protein folding and degradation.

Boschelli F, Golas JM, Petersen R, Lau V, Chen L, Tkach D, Zhao Q, Fruhling DS, Liu H, Nam C, Arndt KT. Boschelli F, et al. Cell Stress Chaperones. 2010 Nov;15(6):913-27. doi: 10.1007/s12192-010-0200-3. Epub 2010 Aug 19. Cell Stress Chaperones. 2010. PMID: 20717760 Free PMC article.

8

Discovery of benzisoxazoles as potent inhibitors of chaperone heat shock protein 90.

Gopalsamy A, Shi M, Golas J, Vogan E, Jacob J, Johnson M, Lee F, Nilakantan R, Petersen R, Svenson K, Chopra R, Tam MS, Wen Y, Ellingboe J, Arndt K, Boschelli F. Gopalsamy A, et al. Among authors: arndt k. J Med Chem. 2008 Feb 14;51(3):373-5. doi: 10.1021/jm701385c. Epub 2008 Jan 16. J Med Chem. 2008. PMID: 18197612

9

Discovery of dibenzo[c,f][2,7]naphthyridines as potent and selective 3-phosphoinositide-dependent kinase-1 inhibitors.

Gopalsamy A, Shi M, Boschelli DH, Williamson R, Olland A, Hu Y, Krishnamurthy G, Han X, Arndt K, Guo B. Gopalsamy A, et al. Among authors: arndt k. J Med Chem. 2007 Nov 15;50(23):5547-9. doi: 10.1021/jm070851i. Epub 2007 Oct 17. J Med Chem. 2007. PMID: 17941624

10

Identification of a conserved sequence motif that promotes Cdc37 and cyclin D1 binding to Cdk4.

Zhao Q, Boschelli F, Caplan AJ, Arndt KT. Zhao Q, et al. J Biol Chem. 2004 Mar 26;279(13):12560-4. doi: 10.1074/jbc.M308242200. Epub 2003 Dec 30. J Biol Chem. 2004. PMID: 14701845 Free article.

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