Grabowski EJ - Search Results

1

Practical asymmetric synthesis of a potent Cathepsin K inhibitor. Efficient palladium removal following Suzuki coupling.

Chen CY, Dagneau P, Grabowski EJ, Oballa R, O'Shea P, Prasit P, Robichaud J, Tillyer R, Wang X. Chen CY, et al. Among authors: grabowski ej. J Org Chem. 2003 Apr 4;68(7):2633-8. doi: 10.1021/jo0205614. J Org Chem. 2003. PMID: 12662032

2

Practical asymmetric synthesis of a potent PDE4 inhibitor via stereoselective enolate alkylation of a chiral aryl-heteroaryl secondary tosylate.

O'Shea PD, Chen CY, Chen W, Dagneau P, Frey LF, Grabowski EJ, Marcantonio KM, Reamer RA, Tan L, Tillyer RD, Roy A, Wang X, Zhao D. O'Shea PD, et al. Among authors: grabowski ej. J Org Chem. 2005 Apr 15;70(8):3021-30. doi: 10.1021/jo048156v. J Org Chem. 2005. PMID: 15822960

3

Practical asymmetric synthesis of a selective endothelin A receptor (ETA) antagonist.

Song ZJ, Zhao M, Frey L, Li J, Tan L, Chen CY, Tschaen DM, Tillyer R, Grabowski EJ, Volante R, Reider PJ, Kato Y, Okada S, Nemoto T, Sato H, Akao A, Mase T. Song ZJ, et al. Among authors: grabowski ej. Org Lett. 2001 Oct 18;3(21):3357-60. doi: 10.1021/ol016601s. Org Lett. 2001. PMID: 11594833

4

Practical synthesis of a potent hepatitis C virus RNA replication inhibitor.

Bio MM, Xu F, Waters M, Williams JM, Savary KA, Cowden CJ, Yang C, Buck E, Song ZJ, Tschaen DM, Volante RP, Reamer RA, Grabowski EJ. Bio MM, et al. Among authors: grabowski ej. J Org Chem. 2004 Sep 17;69(19):6257-66. doi: 10.1021/jo0491096. J Org Chem. 2004. PMID: 15357584

5

Enantioselective acetylide additions: practical syntheses of non-nucleoside reverse transcriptase inhibitors.

Tillyer RD, Grabowski EJ. Tillyer RD, et al. Among authors: grabowski ej. Curr Opin Drug Discov Devel. 1998 Nov;1(3):349-57. Curr Opin Drug Discov Devel. 1998. PMID: 19649809 No abstract available.

6

Synthesis of alpha-amido ketones via organic catalysis: thiazolium-catalyzed cross-coupling of aldehydes with acylimines.

Murry JA, Frantz DE, Soheili A, Tillyer R, Grabowski EJ, Reider PJ. Murry JA, et al. Among authors: grabowski ej. J Am Chem Soc. 2001 Oct 3;123(39):9696-7. doi: 10.1021/ja0165943. J Am Chem Soc. 2001. PMID: 11572700 No abstract available.

7

Asymmetric synthesis of a prostaglandin D2 receptor antagonist.

Campos KR, Journet M, Lee S, Grabowski EJ, Tillyer RD. Campos KR, et al. Among authors: grabowski ej. J Org Chem. 2005 Jan 7;70(1):268-74. doi: 10.1021/jo048305+. J Org Chem. 2005. PMID: 15624932

8

A practical and efficient preparation of the releasable naphthosultam side chain of a novel anti-MRSA carbapenem.

Miller RA, Humphrey GR, Lieberman DR, Ceglia SS, Kennedy DJ, Grabowski EJ, Reider PJ. Miller RA, et al. Among authors: grabowski ej. J Org Chem. 2000 Mar 10;65(5):1399-406. doi: 10.1021/jo991490k. J Org Chem. 2000. PMID: 10814101

9

Stereoselective formation of carbon-carbon bonds via SN2-displacement: synthesis of substituted cycloalkyl[b]indoles.

Hillier MC, Marcoux JF, Zhao D, Grabowski EJ, McKeown AE, Tillyer RD. Hillier MC, et al. Among authors: grabowski ej. J Org Chem. 2005 Oct 14;70(21):8385-94. doi: 10.1021/jo051146p. J Org Chem. 2005. PMID: 16209582

10

An Asymmetric Synthesis of L-694,458, a Human Leukocyte Elastase Inhibitor, via Novel Enzyme Resolution of beta-Lactam Esters.

Cvetovich RJ, Chartrain M, Hartner FW Jr, Roberge C, Amato JS, Grabowski EJ. Cvetovich RJ, et al. Among authors: grabowski ej. J Org Chem. 1996 Sep 20;61(19):6575-6580. doi: 10.1021/jo960618k. J Org Chem. 1996. PMID: 11667523

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