Sbacchi M - Search Results

1

Synthesis, biological evaluation, and receptor docking simulations of 2-[(acylamino)ethyl]-1,4-benzodiazepines as kappa-opioid receptor agonists endowed with antinociceptive and antiamnesic activity.

Anzini M, Canullo L, Braile C, Cappelli A, Gallelli A, Vomero S, Menziani MC, De Benedetti PG, Rizzo M, Collina S, Azzolina O, Sbacchi M, Ghelardini C, Galeotti N. Anzini M, et al. Among authors: sbacchi m. J Med Chem. 2003 Aug 28;46(18):3853-64. doi: 10.1021/jm0307640. J Med Chem. 2003. PMID: 12930147

2

Synthesis, biological evaluation, and quantitative receptor docking simulations of 2-[(acylamino)ethyl]-1,4-benzodiazepines as novel tifluadom-like ligands with high affinity and selectivity for kappa-opioid receptors.

Cappelli A, Anzini M, Vomero S, Menziani MC, De Benedetti PG, Sbacchi M, Clarke GD, Mennuni L. Cappelli A, et al. Among authors: sbacchi m. J Med Chem. 1996 Feb 16;39(4):860-72. doi: 10.1021/jm950423p. J Med Chem. 1996. PMID: 8632410

3

Synthesis and antinociceptive activity of pyrrolidinylnaphthalenes.

Collina S, Azzolina O, Vercesi D, Sbacchi M, Scheideler MA, Barbieri A, Lanza E, Ghislandi V. Collina S, et al. Among authors: sbacchi m. Bioorg Med Chem. 2000 Aug;8(8):1925-30. doi: 10.1016/s0968-0896(00)00117-6. Bioorg Med Chem. 2000. PMID: 11003137

4

Enantiomers of 2-[(Acylamino)ethyl]-1,4-benzodiazepines, potent ligands of kappa-opioid receptor: chiral chromatographic resolution, configurational assignment and biological activity.

Azzolina O, Collina S, Linati L, Anzini M, Cappelli A, Scheideler MA, Sbacchi M. Azzolina O, et al. Among authors: sbacchi m. Chirality. 2001;13(9):606-12. doi: 10.1002/chir.1185. Chirality. 2001. PMID: 11579457

5

Synthesis and antinociceptive activity of chimonanthines and pyrrolidinoindoline-type alkaloids.

Verotta L, Orsini F, Sbacchi M, Scheildler MA, Amador TA, Elisabetsky E. Verotta L, et al. Among authors: sbacchi m. Bioorg Med Chem. 2002 Jul;10(7):2133-42. doi: 10.1016/s0968-0896(02)00078-0. Bioorg Med Chem. 2002. PMID: 11983509

6

Selective kappa-opioid agonists: synthesis and structure-activity relationships of piperidines incorporating on oxo-containing acyl group.

Giardina G, Clarke GD, Dondio G, Petrone G, Sbacchi M, Vecchietti V. Giardina G, et al. Among authors: sbacchi m. J Med Chem. 1994 Oct 14;37(21):3482-91. doi: 10.1021/jm00047a006. J Med Chem. 1994. PMID: 7932577

7

Substituted 1-(aminomethyl)-2-(arylacetyl)-1,2,3,4-tetrahydroisoquinolines: a novel class of very potent antinociceptive agents with varying degrees of selectivity for kappa and mu opioid receptors.

Vecchietti V, Clarke GD, Colle R, Dondio G, Giardina G, Petrone G, Sbacchi M. Vecchietti V, et al. Among authors: sbacchi m. J Med Chem. 1992 Aug 7;35(16):2970-8. doi: 10.1021/jm00094a006. J Med Chem. 1992. PMID: 1323679

8

(1S)-1-(aminomethyl)-2-(arylacetyl)-1,2,3,4-tetrahydroisoquinoline and heterocycle-condensed tetrahydropyridine derivatives: members of a novel class of very potent kappa opioid analgesics.

Vecchietti V, Clarke GD, Colle R, Giardina G, Petrone G, Sbacchi M. Vecchietti V, et al. Among authors: sbacchi m. J Med Chem. 1991 Aug;34(8):2624-33. doi: 10.1021/jm00112a042. J Med Chem. 1991. PMID: 1652025

9

Side-chain lactam-bridge conformational constraints differentiate the activities of salmon and human calcitonins and reveal a new design concept for potent calcitonin analogues.

Taylor JW, Jin QK, Sbacchi M, Wang L, Belfiore P, Garnier M, Kazantzis A, Kapurniotu A, Zaratin PF, Scheideler MA. Taylor JW, et al. Among authors: sbacchi m. J Med Chem. 2002 Feb 28;45(5):1108-21. doi: 10.1021/jm010474o. J Med Chem. 2002. PMID: 11855991

10

Central and peripheral analgesic agents: chemical strategies for limiting brain penetration in kappa-opioid agonists belonging to different chemical classes.

Giardina G, Clarke GD, Grugni M, Sbacchi M, Vecchietti V. Giardina G, et al. Among authors: sbacchi m. Farmaco. 1995 Jun;50(6):405-18. Farmaco. 1995. PMID: 7669179 Review.

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