Baraldi PG - Search Results

1

Asymmetrical nitrido tc-99m heterocomplexes as potential imaging agents for benzodiazepine receptors.

Boschi A, Uccelli L, Duatti A, Bolzati C, Refosco F, Tisato F, Romagnoli R, Baraldi PG, Varani K, Borea PA. Boschi A, et al. Among authors: baraldi pg. Bioconjug Chem. 2003 Nov-Dec;14(6):1279-88. doi: 10.1021/bc034124n. Bioconjug Chem. 2003. PMID: 14624645

2

7-Substituted 5-amino-2-(2-furyl)pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonists: a study on the importance of modifications at the side chain on the activity and solubility.

Baraldi PG, Cacciari B, Romagnoli R, Spalluto G, Monopoli A, Ongini E, Varani K, Borea PA. Baraldi PG, et al. J Med Chem. 2002 Jan 3;45(1):115-26. doi: 10.1021/jm010924c. J Med Chem. 2002. PMID: 11754583

3

Synthesis and biological effects of novel 2-amino-3-naphthoylthiophenes as allosteric enhancers of the A1 adenosine receptor.

Baraldi PG, Romagnoli R, Pavani MG, Nuñez Mdel C, Tabrizi MA, Shryock JC, Leung E, Moorman AR, Uluoglu C, Iannotta V, Merighi S, Borea PA. Baraldi PG, et al. J Med Chem. 2003 Feb 27;46(5):794-809. doi: 10.1021/jm0210212. J Med Chem. 2003. PMID: 12593659

4

Design, synthesis, and biological evaluation of C9- and C2-substituted pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as new A2A and A3 adenosine receptors antagonists.

Baraldi PG, Fruttarolo F, Tabrizi MA, Preti D, Romagnoli R, El-Kashef H, Moorman A, Varani K, Gessi S, Merighi S, Borea PA. Baraldi PG, et al. J Med Chem. 2003 Mar 27;46(7):1229-41. doi: 10.1021/jm021023m. J Med Chem. 2003. PMID: 12646033

5

New strategies for the synthesis of A3 adenosine receptor antagonists.

Baraldi PG, Bovero A, Fruttarolo F, Romagnoli R, Tabrizi MA, Preti D, Varani K, Borea PA, Moorman AR. Baraldi PG, et al. Bioorg Med Chem. 2003 Sep 15;11(19):4161-9. doi: 10.1016/s0968-0896(03)00484-x. Bioorg Med Chem. 2003. PMID: 12951147

6

Design, synthesis, and biological evaluation of new 8-heterocyclic xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists.

Baraldi PG, Tabrizi MA, Preti D, Bovero A, Romagnoli R, Fruttarolo F, Zaid NA, Moorman AR, Varani K, Gessi S, Merighi S, Borea PA. Baraldi PG, et al. J Med Chem. 2004 Mar 11;47(6):1434-47. doi: 10.1021/jm0309654. J Med Chem. 2004. PMID: 14998332

7

Synthesis, radiolabeling, and preliminary biological evaluation of [3H]-1-[(S)-N,O-bis-(isoquinolinesulfonyl)-N-methyl-tyrosyl]-4-(o-tolyl)-piperazine, a potent antagonist radioligand for the P2X7 receptor.

Romagnoli R, Baraldi PG, Pavani MG, Tabrizi MA, Moorman AR, Di Virgilio F, Cattabriga E, Pancaldi C, Gessi S, Borea PA. Romagnoli R, et al. Among authors: baraldi pg. Bioorg Med Chem Lett. 2004 Nov 15;14(22):5709-12. doi: 10.1016/j.bmcl.2004.07.095. Bioorg Med Chem Lett. 2004. PMID: 15482953

8

New pyrrolo[2,1-f]purine-2,4-dione and imidazo[2,1-f]purine-2,4-dione derivatives as potent and selective human A3 adenosine receptor antagonists.

Baraldi PG, Preti D, Tabrizi MA, Fruttarolo F, Romagnoli R, Zaid NA, Moorman AR, Merighi S, Varani K, Borea PA. Baraldi PG, et al. J Med Chem. 2005 Jul 14;48(14):4697-701. doi: 10.1021/jm058008c. J Med Chem. 2005. PMID: 16000006

9

Synthesis and biological characterization of [3H] (2-amino-4,5,6,7-tetrahydrobenzo[b]thiophen-3-yl)-(4-chlorophenyl)-methanone, the first radiolabelled adenosine A1 allosteric enhancer.

Baraldi PG, Pavani MG, Leung E, Moorman AR, Varani K, Vincenzi F, Borea PA, Romagnoli R. Baraldi PG, et al. Bioorg Med Chem Lett. 2006 Mar 1;16(5):1402-4. doi: 10.1016/j.bmcl.2005.11.037. Bioorg Med Chem Lett. 2006. PMID: 16321527

10

Synthesis and biological evaluation of novel 1-deoxy-1-[6-[((hetero)arylcarbonyl)hydrazino]- 9H-purin-9-yl]-N-ethyl-beta-D-ribofuranuronamide derivatives as useful templates for the development of A2B adenosine receptor agonists.

Baraldi PG, Preti D, Tabrizi MA, Fruttarolo F, Romagnoli R, Carrion MD, Cara LC, Moorman AR, Varani K, Borea PA. Baraldi PG, et al. J Med Chem. 2007 Jan 25;50(2):374-80. doi: 10.1021/jm061170a. J Med Chem. 2007. PMID: 17228880

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