Ruiu S - Search Results

1

Synthesis and biological evaluation of 1,8-naphthyridin-4(1H)-on-3-carboxamide derivatives as new ligands of cannabinoid receptors.

Ferrarini PL, Calderone V, Cavallini T, Manera C, Saccomanni G, Pani L, Ruiu S, Gessa GL. Ferrarini PL, et al. Among authors: ruiu s. Bioorg Med Chem. 2004 Apr 15;12(8):1921-33. doi: 10.1016/j.bmc.2004.01.035. Bioorg Med Chem. 2004. PMID: 15051060

2

Tricyclic pyrazoles. Part 2: Synthesis and biological evaluation of novel 4,5-dihydro-1H-benzo[g]indazole-based ligands for cannabinoid receptors.

Murineddu G, Ruiu S, Mussinu JM, Loriga G, Grella GE, Carai MA, Lazzari P, Pani L, Pinna GA. Murineddu G, et al. Among authors: ruiu s. Bioorg Med Chem. 2005 May 2;13(9):3309-20. doi: 10.1016/j.bmc.2005.02.032. Bioorg Med Chem. 2005. PMID: 15809166

3

Tricyclic pyrazoles. 3. Synthesis, biological evaluation, and molecular modeling of analogues of the cannabinoid antagonist 8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide.

Murineddu G, Ruiu S, Loriga G, Manca I, Lazzari P, Reali R, Pani L, Toma L, Pinna GA. Murineddu G, et al. Among authors: ruiu s. J Med Chem. 2005 Nov 17;48(23):7351-62. doi: 10.1021/jm050317f. J Med Chem. 2005. PMID: 16279795

A series of analogues of 8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 4a (NESS 0327) (Ruiu, S.; Pinna, G. A.; Marchese, G.; Mussinu, J. M.; Saba, P.; Tambaro, S.; Casti, P.; Vargiu, R.; …

A series of analogues of 8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxam …

4

Tricyclic pyrazoles. 4. Synthesis and biological evaluation of analogues of the robust and selective CB2 cannabinoid ligand 1-(2',4'-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide.

Murineddu G, Lazzari P, Ruiu S, Sanna A, Loriga G, Manca I, Falzoi M, Dessì C, Curzu MM, Chelucci G, Pani L, Pinna GA. Murineddu G, et al. Among authors: ruiu s. J Med Chem. 2006 Dec 14;49(25):7502-12. doi: 10.1021/jm060920d. J Med Chem. 2006. PMID: 17149879

5

Tricyclic pyrazoles. Part 1: synthesis and biological evaluation of novel 1,4-dihydroindeno[1,2-c]pyrazol-based ligands for CB1and CB2 cannabinoid receptors.

Mussinu JM, Ruiu S, Mulè AC, Pau A, Carai MA, Loriga G, Murineddu G, Pinna GA. Mussinu JM, et al. Among authors: ruiu s. Bioorg Med Chem. 2003 Jan 17;11(2):251-63. doi: 10.1016/s0968-0896(02)00319-x. Bioorg Med Chem. 2003. PMID: 12470719

6

3-{2-[Bis-(4-fluorophenyl)methoxy]ethyl}-6-substituted-3,6-diazabicyclo[3.1.1]heptanes as novel potent dopamine uptake inhibitors.

Loriga G, Ruiu S, Manca I, Murineddu G, Dessi C, Pani L, Pinna GA. Loriga G, et al. Among authors: ruiu s. Bioorg Med Chem. 2007 Jun 1;15(11):3748-55. doi: 10.1016/j.bmc.2007.03.035. Epub 2007 Mar 16. Bioorg Med Chem. 2007. PMID: 17399987

7

Tricyclic Pyrazoles. Part 5. Novel 1,4-Dihydroindeno[1,2-c]pyrazole CB2 Ligands Using Molecular Hybridization Based on Scaffold Hopping.

Murineddu G, Asproni B, Ruiu S, Deligia F, Falzoi M, Pau A, Thomas BF, Zhang Y, Pinna GA, Pani L, Lazzari P. Murineddu G, et al. Among authors: ruiu s. Open Med Chem J. 2012;6:1-14. doi: 10.2174/1874104501206010001. Epub 2012 May 17. Open Med Chem J. 2012. PMID: 22876271 Free PMC article.

8

Differential distribution of functional cannabinoid CB1 receptors in the mouse gastroenteric tract.

Casu MA, Porcella A, Ruiu S, Saba P, Marchese G, Carai MA, Reali R, Gessa GL, Pani L. Casu MA, et al. Among authors: ruiu s. Eur J Pharmacol. 2003 Jan 10;459(1):97-105. doi: 10.1016/s0014-2999(02)02830-3. Eur J Pharmacol. 2003. PMID: 12505538

9

Synthesis and characterization of NESS 0327: a novel putative antagonist of the CB1 cannabinoid receptor.

Ruiu S, Pinna GA, Marchese G, Mussinu JM, Saba P, Tambaro S, Casti P, Vargiu R, Pani L. Ruiu S, et al. J Pharmacol Exp Ther. 2003 Jul;306(1):363-70. doi: 10.1124/jpet.103.049924. Epub 2003 Mar 27. J Pharmacol Exp Ther. 2003. PMID: 12663689

10

Synthesis and in vitro Evaluation of Trifluoroethylamine Analogues of Enkephalins.

Sinisi R, Ghilardi A, Ruiu S, Lazzari P, Malpezzi L, Sani M, Pani L, Zanda M. Sinisi R, et al. Among authors: ruiu s. ChemMedChem. 2009 Sep;4(9):1416-20. doi: 10.1002/cmdc.200900158. ChemMedChem. 2009. PMID: 19533725 No abstract available.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

64 results

Search Page

Filters