van Rijn RM - Search Results

1

Synthesis and structure-activity relationships of indole and benzimidazole piperazines as histamine H(4) receptor antagonists.

Terzioglu N, van Rijn RM, Bakker RA, De Esch IJ, Leurs R. Terzioglu N, et al. Among authors: van rijn rm. Bioorg Med Chem Lett. 2004 Nov 1;14(21):5251-6. doi: 10.1016/j.bmcl.2004.08.035. Bioorg Med Chem Lett. 2004. PMID: 15454206

2

Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.

Lim HD, van Rijn RM, Ling P, Bakker RA, Thurmond RL, Leurs R. Lim HD, et al. Among authors: van rijn rm. J Pharmacol Exp Ther. 2005 Sep;314(3):1310-21. doi: 10.1124/jpet.105.087965. Epub 2005 Jun 9. J Pharmacol Exp Ther. 2005. PMID: 15947036

3

Discovery of naturally occurring splice variants of the rat histamine H3 receptor that act as dominant-negative isoforms.

Bakker RA, Lozada AF, van Marle A, Shenton FC, Drutel G, Karlstedt K, Hoffmann M, Lintunen M, Yamamoto Y, van Rijn RM, Chazot PL, Panula P, Leurs R. Bakker RA, et al. Among authors: van rijn rm, van marle a. Mol Pharmacol. 2006 Apr;69(4):1194-206. doi: 10.1124/mol.105.019299. Epub 2006 Jan 13. Mol Pharmacol. 2006. PMID: 16415177

4

Oligomerization of recombinant and endogenously expressed human histamine H(4) receptors.

van Rijn RM, Chazot PL, Shenton FC, Sansuk K, Bakker RA, Leurs R. van Rijn RM, et al. Mol Pharmacol. 2006 Aug;70(2):604-15. doi: 10.1124/mol.105.020818. Epub 2006 Apr 27. Mol Pharmacol. 2006. PMID: 16645125

5

Cloning and characterization of dominant negative splice variants of the human histamine H4 receptor.

van Rijn RM, van Marle A, Chazot PL, Langemeijer E, Qin Y, Shenton FC, Lim HD, Zuiderveld OP, Sansuk K, Dy M, Smit MJ, Tensen CP, Bakker RA, Leurs R. van Rijn RM, et al. Among authors: van marle a. Biochem J. 2008 Aug 15;414(1):121-31. doi: 10.1042/BJ20071583. Biochem J. 2008. PMID: 18452403

6

A Novel Mitragynine Analog with Low-Efficacy Mu Opioid Receptor Agonism Displays Antinociception with Attenuated Adverse Effects.

Chakraborty S, DiBerto JF, Faouzi A, Bernhard SM, Gutridge AM, Ramsey S, Zhou Y, Provasi D, Nuthikattu N, Jilakara R, Nelson MNF, Asher WB, Eans SO, Wilson LL, Chintala SM, Filizola M, van Rijn RM, Margolis EB, Roth BL, McLaughlin JP, Che T, Sames D, Javitch JA, Majumdar S. Chakraborty S, et al. Among authors: van rijn rm. J Med Chem. 2021 Sep 23;64(18):13873-13892. doi: 10.1021/acs.jmedchem.1c01273. Epub 2021 Sep 10. J Med Chem. 2021. PMID: 34505767 Free PMC article.

7

Modified Akuamma Alkaloids with Increased Potency at the Mu-opioid Receptor.

Hennessy MR, Gutridge AM, French AR, Rhoda ES, Meqbil YJ, Gill M, Kashyap Y, Appourchaux K, Paul B, Wang ZJ, van Rijn RM, Riley AP. Hennessy MR, et al. Among authors: van rijn rm. J Med Chem. 2023 Mar 9;66(5):3312-3326. doi: 10.1021/acs.jmedchem.2c01707. Epub 2023 Feb 24. J Med Chem. 2023. PMID: 36827198 Free PMC article.

8

Optimization of a 1,3,4-oxadiazole series for inhibition of Ca²⁺/calmodulin-stimulated activity of adenylyl cyclases 1 and 8 for the treatment of chronic pain.

Kaur J, Soto-Velasquez M, Ding Z, Ghanbarpour A, Lill MA, van Rijn RM, Watts VJ, Flaherty DP. Kaur J, et al. Among authors: van rijn rm. Eur J Med Chem. 2019 Jan 15;162:568-585. doi: 10.1016/j.ejmech.2018.11.036. Epub 2018 Nov 16. Eur J Med Chem. 2019. PMID: 30472604 Free PMC article.

9

Opioids and Their Receptors: Present and Emerging Concepts in Opioid Drug Discovery II.

Van Rijn RM, Spetea M. Van Rijn RM, et al. Molecules. 2022 May 13;27(10):3140. doi: 10.3390/molecules27103140. Molecules. 2022. PMID: 35630616 Free PMC article.

10

Dual efficacy of delta opioid receptor-selective ligands for ethanol drinking and anxiety.

van Rijn RM, Brissett DI, Whistler JL. van Rijn RM, et al. J Pharmacol Exp Ther. 2010 Oct;335(1):133-9. doi: 10.1124/jpet.110.170969. Epub 2010 Jul 6. J Pharmacol Exp Ther. 2010. PMID: 20605909 Free PMC article.

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