van der Veken P - Search Results

1

Development of a novel chemical probe for the selective enrichment of phosphorylated serine- and threonine-containing peptides.

van der Veken P, Dirksen EH, Ruijter E, Elgersma RC, Heck AJ, Rijkers DT, Slijper M, Liskamp RM. van der Veken P, et al. Chembiochem. 2005 Dec;6(12):2271-80. doi: 10.1002/cbic.200500209. Chembiochem. 2005. PMID: 16254931

2

Repositioning the substrate activity screening (SAS) approach as a fragment-based method for identification of weak binders.

Gladysz R, Cleenewerck M, Joossens J, Lambeir AM, Augustyns K, Van der Veken P. Gladysz R, et al. Among authors: van der veken p. Chembiochem. 2014 Oct 13;15(15):2238-47. doi: 10.1002/cbic.201402192. Epub 2014 Aug 25. Chembiochem. 2014. PMID: 25154878

3

Inhibitors of dipeptidyl peptidase 8 and dipeptidyl peptidase 9. Part 2: isoindoline containing inhibitors.

Van Goethem S, Van der Veken P, Dubois V, Soroka A, Lambeir AM, Chen X, Haemers A, Scharpé S, De Meester I, Augustyns K. Van Goethem S, et al. Among authors: van der veken p. Bioorg Med Chem Lett. 2008 Jul 15;18(14):4159-62. doi: 10.1016/j.bmcl.2008.05.079. Epub 2008 May 24. Bioorg Med Chem Lett. 2008. PMID: 18556198

4

Development of potent and selective dipeptidyl peptidase II inhibitors.

Senten K, Van der Veken P, Bal G, De Meester I, Lambeir AM, Scharpé S, Bauvois B, Haemers A, Augustyns K. Senten K, et al. Among authors: van der veken p. Bioorg Med Chem Lett. 2002 Oct 21;12(20):2825-8. doi: 10.1016/s0960-894x(02)00603-0. Bioorg Med Chem Lett. 2002. PMID: 12270155

5

Structure-activity relationship studies on isoindoline inhibitors of dipeptidyl peptidases 8 and 9 (DPP8, DPP9): is DPP8-selectivity an attainable goal?

Van Goethem S, Matheeussen V, Joossens J, Lambeir AM, Chen X, De Meester I, Haemers A, Augustyns K, Van der Veken P. Van Goethem S, et al. Among authors: van der veken p. J Med Chem. 2011 Aug 25;54(16):5737-46. doi: 10.1021/jm200383j. Epub 2011 Aug 2. J Med Chem. 2011. PMID: 21711053

6

P2-substituted N-acylprolylpyrrolidine inhibitors of prolyl oligopeptidase: biochemical evaluation, binding mode determination, and assessment in a cellular model of synucleinopathy.

Van der Veken P, Fülöp V, Rea D, Gerard M, Van Elzen R, Joossens J, Cheng JD, Baekelandt V, De Meester I, Lambeir AM, Augustyns K. Van der Veken P, et al. Among authors: van elzen r. J Med Chem. 2012 Nov 26;55(22):9856-67. doi: 10.1021/jm301060g. Epub 2012 Nov 13. J Med Chem. 2012. PMID: 23121075

7

Glutathione-like tripeptides as inhibitors of glutathionylspermidine synthetase. Part 2: substitution of the glycine part.

Amssoms K, Oza SL, Augustyns K, Yamani A, Lambeir AM, Bal G, Van der Veken P, Fairlamb AH, Haemers A. Amssoms K, et al. Among authors: van der veken p. Bioorg Med Chem Lett. 2002 Oct 7;12(19):2703-5. doi: 10.1016/s0960-894x(02)00538-3. Bioorg Med Chem Lett. 2002. PMID: 12217358

8

Rapid parallel synthesis of dipeptide diphenyl phosphonate esters as inhibitors of dipeptidyl peptidases.

Senten K, Daniëls L, Van der Veken P, De Meester I, Lambeir AM, Scharpé S, Haemers A, Augustyns K. Senten K, et al. Among authors: van der veken p. J Comb Chem. 2003 May-Jun;5(3):336-44. doi: 10.1021/cc020096o. J Comb Chem. 2003. PMID: 12739951

9

Design, synthesis, and SAR of potent and selective dipeptide-derived inhibitors for dipeptidyl peptidases.

Senten K, Van der Veken P, De Meester I, Lambeir AM, Scharpé S, Haemers A, Augustyns K. Senten K, et al. Among authors: van der veken p. J Med Chem. 2003 Nov 6;46(23):5005-14. doi: 10.1021/jm0308803. J Med Chem. 2003. PMID: 14584950

10

Development of irreversible diphenyl phosphonate inhibitors for urokinase plasminogen activator.

Joossens J, Van der Veken P, Lambeir AM, Augustyns K, Haemers A. Joossens J, et al. Among authors: van der veken p. J Med Chem. 2004 May 6;47(10):2411-3. doi: 10.1021/jm0499209. J Med Chem. 2004. PMID: 15115382

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