Hales NJ - Search Results

1

New carbon-linked azole oxazolidinones with improved potency and pharmacokinetics.

Hauck SI, Cederberg C, Doucette A, Grosser L, Hales NJ, Poon G, Gravestock MB. Hauck SI, et al. Among authors: hales nj. Bioorg Med Chem Lett. 2007 Jan 15;17(2):337-40. doi: 10.1016/j.bmcl.2006.10.063. Epub 2006 Oct 26. Bioorg Med Chem Lett. 2007. PMID: 17095223

2

Identification of 4-substituted 1,2,3-triazoles as novel oxazolidinone antibacterial agents with reduced activity against monoamine oxidase A.

Reck F, Zhou F, Girardot M, Kern G, Eyermann CJ, Hales NJ, Ramsay RR, Gravestock MB. Reck F, et al. Among authors: hales nj. J Med Chem. 2005 Jan 27;48(2):499-506. doi: 10.1021/jm0400810. J Med Chem. 2005. PMID: 15658863

3

Pyrrolamide DNA gyrase inhibitors: fragment-based nuclear magnetic resonance screening to identify antibacterial agents.

Eakin AE, Green O, Hales N, Walkup GK, Bist S, Singh A, Mullen G, Bryant J, Embrey K, Gao N, Breeze A, Timms D, Andrews B, Uria-Nickelsen M, Demeritt J, Loch JT 3rd, Hull K, Blodgett A, Illingworth RN, Prince B, Boriack-Sjodin PA, Hauck S, MacPherson LJ, Ni H, Sherer B. Eakin AE, et al. Antimicrob Agents Chemother. 2012 Mar;56(3):1240-6. doi: 10.1128/AAC.05485-11. Epub 2011 Dec 19. Antimicrob Agents Chemother. 2012. PMID: 22183167 Free PMC article.

4

Small-molecule androgen receptor downregulators as an approach to treatment of advanced prostate cancer.

Bradbury RH, Hales NJ, Rabow AA, Walker GE, Acton DG, Andrews DM, Ballard P, Brooks NA, Colclough N, Girdwood A, Hancox UJ, Jones O, Jude D, Loddick SA, Mortlock AA. Bradbury RH, et al. Among authors: hales nj. Bioorg Med Chem Lett. 2011 Sep 15;21(18):5442-5. doi: 10.1016/j.bmcl.2011.06.122. Epub 2011 Jul 2. Bioorg Med Chem Lett. 2011. PMID: 21782422

5

Novel inhibitors of prolyl 4-hydroxylase. 5. The intriguing structure-activity relationships seen with 2,2'-bipyridine and its 5,5'-dicarboxylic acid derivatives.

Hales NJ, Beattie JF. Hales NJ, et al. J Med Chem. 1993 Nov 26;36(24):3853-8. doi: 10.1021/jm00076a014. J Med Chem. 1993. PMID: 8254616

6

Novel inhibitors of prolyl 4-hydroxylase. 3. Inhibition by the substrate analogue N-oxaloglycine and its derivatives.

Cunliffe CJ, Franklin TJ, Hales NJ, Hill GB. Cunliffe CJ, et al. Among authors: hales nj. J Med Chem. 1992 Jul 10;35(14):2652-8. doi: 10.1021/jm00092a016. J Med Chem. 1992. PMID: 1321909

7

Kinetic and structural characteristics of the inhibition of enoyl (acyl carrier protein) reductase by triclosan.

Ward WH, Holdgate GA, Rowsell S, McLean EG, Pauptit RA, Clayton E, Nichols WW, Colls JG, Minshull CA, Jude DA, Mistry A, Timms D, Camble R, Hales NJ, Britton CJ, Taylor IW. Ward WH, et al. Among authors: hales nj. Biochemistry. 1999 Sep 21;38(38):12514-25. doi: 10.1021/bi9907779. Biochemistry. 1999. PMID: 10493822

8

Approaches to the design of anti-fibrotic drugs.

Franklin TJ, Hales NJ, Johnstone D, Morris WB, Cunliffe CJ, Millest AJ, Hill GB. Franklin TJ, et al. Among authors: hales nj. Biochem Soc Trans. 1991 Nov;19(4):812-5. doi: 10.1042/bst0190812. Biochem Soc Trans. 1991. PMID: 1665444 No abstract available.

9

The application of polymer-bound carbonylcobalt(0) species in linker chemistry and catalysis.

Comely AC, Gibson SE, Hales NJ, Johnstone C, Stevenazzi A. Comely AC, et al. Among authors: hales nj. Org Biomol Chem. 2003 Jun 7;1(11):1959-68. doi: 10.1039/b303208f. Org Biomol Chem. 2003. PMID: 12945780

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