Melchiorre C - Search Results

1

Synthesis and alpha(1)-adrenoceptor antagonist activity of derivatives and isosters of the furan portion of (+)-cyclazosin.

Sagratini G, Angeli P, Buccioni M, Gulini U, Marucci G, Melchiorre C, Leonardi A, Poggesi E, Giardinà D. Sagratini G, et al. Among authors: melchiorre c. Bioorg Med Chem. 2007 Mar 15;15(6):2334-45. doi: 10.1016/j.bmc.2007.01.028. Epub 2007 Jan 19. Bioorg Med Chem. 2007. PMID: 17276073

2

Structure--activity relationships among novel phenoxybenzamine-related beta-chloroethylamines.

Giardinà D, Crucianelli M, Angeli P, Buccioni M, Gulini U, Marucci G, Sagratini G, Melchiorre C. Giardinà D, et al. Among authors: melchiorre c. Bioorg Med Chem. 2002 May;10(5):1291-303. doi: 10.1016/s0968-0896(01)00395-9. Bioorg Med Chem. 2002. PMID: 11886792

3

Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes.

Quaglia W, Pigini M, Piergentili A, Giannella M, Gentili F, Marucci G, Carrieri A, Carotti A, Poggesi E, Leonardi A, Melchiorre C. Quaglia W, et al. Among authors: melchiorre c. J Med Chem. 2002 Apr 11;45(8):1633-43. doi: 10.1021/jm011066n. J Med Chem. 2002. PMID: 11931617

4

Rosini M, Antonello A, Cavalli A, Bolognesi ML, Minarini A, Marucci G, Poggesi E, Leonardi A, Melchiorre C. Rosini M, et al. Among authors: melchiorre c. J Med Chem. 2003 Nov 6;46(23):4895-903. doi: 10.1021/jm030952q. J Med Chem. 2003. PMID: 14584940

5

Absolute configuration of the alpha (1B)-adrenoceptor antagonist (+)-cyclazosin.

Giardinà D, Sagratini G, Grelli M, Gulini U, Melchiorre C, Antolini L. Giardinà D, et al. Among authors: melchiorre c. Farmaco. 2004 Dec;59(12):965-9. doi: 10.1016/j.farmac.2004.07.013. Farmaco. 2004. PMID: 15598431

6

Design, synthesis, and biological evaluation of prazosin-related derivatives as multipotent compounds.

Antonello A, Hrelia P, Leonardi A, Marucci G, Rosini M, Tarozzi A, Tumiatti V, Melchiorre C. Antonello A, et al. Among authors: melchiorre c. J Med Chem. 2005 Jan 13;48(1):28-31. doi: 10.1021/jm049153d. J Med Chem. 2005. PMID: 15633998

7

(+)-Cyclazosin, a selective alpha1B-adrenoceptor antagonist: functional evaluation in rat and rabbit tissues.

Marucci G, Angeli P, Buccioni M, Gulini U, Melchiorre C, Sagratini G, Testa R, Giardinà D. Marucci G, et al. Among authors: melchiorre c. Eur J Pharmacol. 2005 Oct 17;522(1-3):100-7. doi: 10.1016/j.ejphar.2005.08.044. Epub 2005 Oct 6. Eur J Pharmacol. 2005. PMID: 16213480

8

Structure-activity relationships of methoctramine-related polyamines as muscarinic antagonist: effect of replacing the inner polymethylene chain with cyclic moieties.

Tumiatti V, Minarini A, Milelli A, Rosini M, Buccioni M, Marucci G, Ghelardini C, Bellucci C, Melchiorre C. Tumiatti V, et al. Among authors: melchiorre c. Bioorg Med Chem. 2007 Mar 15;15(6):2312-21. doi: 10.1016/j.bmc.2007.01.022. Epub 2007 Jan 19. Bioorg Med Chem. 2007. PMID: 17276075

9

Doxazosin-related alpha1-adrenoceptor antagonists with prostate antitumor activity.

Giardinà D, Martarelli D, Sagratini G, Angeli P, Ballinari D, Gulini U, Melchiorre C, Poggesi E, Pompei P. Giardinà D, et al. Among authors: melchiorre c. J Med Chem. 2009 Aug 13;52(15):4951-4. doi: 10.1021/jm8016046. J Med Chem. 2009. PMID: 19719240

10

Synthesis and α1-adrenoceptor antagonist activity of tamsulosin analogues.

Sagratini G, Angeli P, Buccioni M, Gulini U, Marucci G, Melchiorre C, Poggesi E, Giardinà D. Sagratini G, et al. Among authors: melchiorre c. Eur J Med Chem. 2010 Dec;45(12):5800-7. doi: 10.1016/j.ejmech.2010.09.042. Epub 2010 Sep 25. Eur J Med Chem. 2010. PMID: 20934789

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

173 results

Search Page

Filters