Yunes RA - Search Results

1

Discovery of structurally diverse HIV-1 integrase inhibitors based on a chalcone pharmacophore.

Deng J, Sanchez T, Al-Mawsawi LQ, Dayam R, Yunes RA, Garofalo A, Bolger MB, Neamati N. Deng J, et al. Among authors: yunes ra. Bioorg Med Chem. 2007 Jul 15;15(14):4985-5002. doi: 10.1016/j.bmc.2007.04.041. Epub 2007 Apr 25. Bioorg Med Chem. 2007. PMID: 17502148

2

Synthesis and pharmacological activity of chalcones derived from 2,4,6-trimethoxyacetophenone in RAW 264.7 cells stimulated by LPS: quantitative structure-activity relationships.

Chiaradia LD, dos Santos R, Vitor CE, Vieira AA, Leal PC, Nunes RJ, Calixto JB, Yunes RA. Chiaradia LD, et al. Among authors: yunes ra. Bioorg Med Chem. 2008 Jan 15;16(2):658-67. doi: 10.1016/j.bmc.2007.10.039. Epub 2007 Oct 18. Bioorg Med Chem. 2008. PMID: 17988874

3

Trimethoxy-chalcone derivatives inhibit growth of Leishmania braziliensis: synthesis, biological evaluation, molecular modeling and structure-activity relationship (SAR).

Bello ML, Chiaradia LD, Dias LR, Pacheco LK, Stumpf TR, Mascarello A, Steindel M, Yunes RA, Castro HC, Nunes RJ, Rodrigues CR. Bello ML, et al. Among authors: yunes ra. Bioorg Med Chem. 2011 Aug 15;19(16):5046-52. doi: 10.1016/j.bmc.2011.06.023. Epub 2011 Jun 21. Bioorg Med Chem. 2011. PMID: 21757358

4

Structure-activity relationships for a collection of structurally diverse inhibitors of purine nucleoside phosphorylase.

Andricopulo AD, Yunes RA. Andricopulo AD, et al. Among authors: yunes ra. Chem Pharm Bull (Tokyo). 2001 Jan;49(1):10-7. doi: 10.1248/cpb.49.10. Chem Pharm Bull (Tokyo). 2001. PMID: 11201210 Free article.

5

Synthesis of chalcone analogues with increased antileishmanial activity.

Boeck P, Bandeira Falcão CA, Leal PC, Yunes RA, Filho VC, Torres-Santos EC, Rossi-Bergmann B. Boeck P, et al. Among authors: yunes ra. Bioorg Med Chem. 2006 Mar 1;14(5):1538-45. doi: 10.1016/j.bmc.2005.10.005. Epub 2005 Dec 28. Bioorg Med Chem. 2006. PMID: 16386424

6

Synthetic chalcones as efficient inhibitors of Mycobacterium tuberculosis protein tyrosine phosphatase PtpA.

Chiaradia LD, Mascarello A, Purificação M, Vernal J, Cordeiro MN, Zenteno ME, Villarino A, Nunes RJ, Yunes RA, Terenzi H. Chiaradia LD, et al. Among authors: yunes ra. Bioorg Med Chem Lett. 2008 Dec 1;18(23):6227-30. doi: 10.1016/j.bmcl.2008.09.105. Epub 2008 Oct 5. Bioorg Med Chem Lett. 2008. PMID: 18930396

7

Inhibition of Mycobacterium tuberculosis tyrosine phosphatase PtpA by synthetic chalcones: kinetics, molecular modeling, toxicity and effect on growth.

Mascarello A, Chiaradia LD, Vernal J, Villarino A, Guido RV, Perizzolo P, Poirier V, Wong D, Martins PG, Nunes RJ, Yunes RA, Andricopulo AD, Av-Gay Y, Terenzi H. Mascarello A, et al. Among authors: yunes ra. Bioorg Med Chem. 2010 Jun 1;18(11):3783-9. doi: 10.1016/j.bmc.2010.04.051. Epub 2010 Apr 21. Bioorg Med Chem. 2010. PMID: 20462762 Free article.

8

Synthesis, biological evaluation, and molecular modeling of chalcone derivatives as potent inhibitors of Mycobacterium tuberculosis protein tyrosine phosphatases (PtpA and PtpB).

Chiaradia LD, Martins PG, Cordeiro MN, Guido RV, Ecco G, Andricopulo AD, Yunes RA, Vernal J, Nunes RJ, Terenzi H. Chiaradia LD, et al. Among authors: yunes ra. J Med Chem. 2012 Jan 12;55(1):390-402. doi: 10.1021/jm2012062. Epub 2011 Dec 20. J Med Chem. 2012. PMID: 22136336

9

Activity of novel quinoxaline-derived chalcones on in vitro glioma cell proliferation.

Mielcke TR, Mascarello A, Filippi-Chiela E, Zanin RF, Lenz G, Leal PC, Chiaradia LD, Yunes RA, Nunes RJ, Battastini AM, Morrone FB, Campos MM. Mielcke TR, et al. Among authors: yunes ra. Eur J Med Chem. 2012 Feb;48:255-64. doi: 10.1016/j.ejmech.2011.12.023. Epub 2011 Dec 22. Eur J Med Chem. 2012. PMID: 22209415

10

Symmetric bis-chalcones as a new type of breast cancer resistance protein inhibitors with a mechanism different from that of chromones.

Winter E, Devantier Neuenfeldt P, Chiaradia-Delatorre LD, Gauthier C, Yunes RA, Nunes RJ, Creczynski-Pasa TB, Di Pietro A. Winter E, et al. Among authors: yunes ra. J Med Chem. 2014 Apr 10;57(7):2930-41. doi: 10.1021/jm401879z. Epub 2014 Mar 24. J Med Chem. 2014. PMID: 24611893

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