Mayorov AV - Search Results

1

Structure-activity relationships of cyclic lactam analogues of alpha-melanocyte-stimulating hormone (alpha-MSH) targeting the human melanocortin-3 receptor.

Mayorov AV, Cai M, Palmer ES, Dedek MM, Cain JP, Van Scoy AR, Tan B, Vagner J, Trivedi D, Hruby VJ. Mayorov AV, et al. J Med Chem. 2008 Jan 24;51(2):187-95. doi: 10.1021/jm070461w. Epub 2007 Dec 19. J Med Chem. 2008. PMID: 18088090 Free PMC article.

2

Novel 3D pharmacophore of alpha-MSH/gamma-MSH hybrids leads to selective human MC1R and MC3R analogues.

Cai M, Mayorov AV, Cabello C, Stankova M, Trivedi D, Hruby VJ. Cai M, et al. Among authors: mayorov av. J Med Chem. 2005 Mar 24;48(6):1839-48. doi: 10.1021/jm049579s. J Med Chem. 2005. PMID: 15771429

3

Design of novel melanotropin agonists and antagonists with high potency and selectivity for human melanocortin receptors.

Cai M, Mayorov AV, Ying J, Stankova M, Trivedi D, Cabello C, Hruby VJ. Cai M, et al. Among authors: mayorov av. Peptides. 2005 Aug;26(8):1481-5. doi: 10.1016/j.peptides.2005.03.020. Peptides. 2005. PMID: 15876475 Review.

4

Structure-activity studies of new melanocortin peptides containing an aromatic amino acid at the N-terminal position.

Grieco P, Cai M, Mayorov AV, Trivedi D, Hruby VJ. Grieco P, et al. Among authors: mayorov av. Peptides. 2006 Feb;27(2):472-81. doi: 10.1016/j.peptides.2005.01.032. Epub 2005 Nov 21. Peptides. 2006. PMID: 16303211 Free PMC article.

5

Development of cyclic gamma-MSH analogues with selective hMC3R agonist and hMC3R/hMC5R antagonist activities.

Mayorov AV, Cai M, Chandler KB, Petrov RR, Van Scoy AR, Yu Z, Tanaka DK, Trivedi D, Hruby VJ. Mayorov AV, et al. J Med Chem. 2006 Mar 23;49(6):1946-52. doi: 10.1021/jm0510326. J Med Chem. 2006. PMID: 16539382 Free PMC article.

6

Effects of macrocycle size and rigidity on melanocortin receptor-1 and -5 selectivity in cyclic lactam alpha-melanocyte-stimulating hormone analogs.

Mayorov AV, Han SY, Cai M, Hammer MR, Trivedi D, Hruby VJ. Mayorov AV, et al. Chem Biol Drug Des. 2006 May;67(5):329-35. doi: 10.1111/j.1747-0285.2006.00383.x. Chem Biol Drug Des. 2006. PMID: 16784457 Free PMC article.

7

Design, synthesis, and biological evaluation of a new class of small molecule peptide mimetics targeting the melanocortin receptors.

Cain JP, Mayorov AV, Cai M, Wang H, Tan B, Chandler K, Lee Y, Petrov RR, Trivedi D, Hruby VJ. Cain JP, et al. Among authors: mayorov av. Bioorg Med Chem Lett. 2006 Oct 15;16(20):5462-7. doi: 10.1016/j.bmcl.2006.07.015. Epub 2006 Aug 22. Bioorg Med Chem Lett. 2006. PMID: 16931008 Free PMC article.

8

Novel selective human melanocortin-3 receptor ligands: use of the 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-one (Aba) scaffold.

Ballet S, Mayorov AV, Cai M, Tymecka D, Chandler KB, Palmer ES, Rompaey KV, Misicka A, Tourwé D, Hruby VJ. Ballet S, et al. Among authors: mayorov av. Bioorg Med Chem Lett. 2007 May 1;17(9):2492-8. doi: 10.1016/j.bmcl.2007.02.020. Epub 2007 Feb 9. Bioorg Med Chem Lett. 2007. PMID: 17314042 Free PMC article.

9

Design, synthesis and biological evaluation of ligands selective for the melanocortin-3 receptor.

Hruby VJ, Cai M, Cain JP, Mayorov AV, Dedek MM, Trivedi D. Hruby VJ, et al. Among authors: mayorov av. Curr Top Med Chem. 2007;7(11):1107-19. doi: 10.2174/156802607780906645. Curr Top Med Chem. 2007. PMID: 17584128 Free PMC article. Review.

10

Melanocortin receptors, melanotropic peptides and penile erection.

King SH, Mayorov AV, Balse-Srinivasan P, Hruby VJ, Vanderah TW, Wessells H. King SH, et al. Among authors: mayorov av. Curr Top Med Chem. 2007;7(11):1098-1106. Curr Top Med Chem. 2007. PMID: 17584130 Free PMC article.

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