Staples DJ - Search Results

1

Exploiting the molecular template of angiotensinogen in the discovery and design of peptidyl, pseudopeptidyl and peptidimimetic inhibitors of human renin: a structure-activity perspective.

Sawyer TK, Hester JB, Schostarez HJ, Thaisrivongs S, Bundy GL, Liu L, Bradford VS, De Vaux AE, Staples DJ, Maggiora LL, et al. Sawyer TK, et al. Among authors: staples dj. Adv Exp Med Biol. 1991;306:307-23. doi: 10.1007/978-1-4684-6012-4_37. Adv Exp Med Biol. 1991. PMID: 1812721 Review. No abstract available.

2

Substrate specificity and inhibitor structure-activity relationships of recombinant human renin: implications in the in vivo evaluation of renin inhibitors.

Evans DB, Cornette JC, Sawyer TK, Staples DJ, de Vaux AE, Sharma SK. Evans DB, et al. Among authors: staples dj. Biotechnol Appl Biochem. 1990 Apr;12(2):161-75. Biotechnol Appl Biochem. 1990. PMID: 2184838

3

Design, structure-activity, and molecular modeling studies of potent renin inhibitory peptides having N-terminal Nin-For-Trp (Ftr): angiotensinogen congeners modified by P1-P1' Phe-Phe, Sta, Leu psi[CH(OH)CH2]Val or leu psi[CH2NH]Val substitutions.

Sawyer TK, Pals DT, Mao B, Staples DJ, de Vaux AE, Maggiora LL, Affholter JA, Kati W, Duchamp D, Hester JB, et al. Sawyer TK, et al. Among authors: staples dj. J Med Chem. 1988 Jan;31(1):18-30. doi: 10.1021/jm00396a006. J Med Chem. 1988. PMID: 3275777

4

HIV protease (HIV PR) inhibitor structure-activity-selectivity, and active site molecular modeling of high affinity Leu [CH(OH)CH2]Val modified viral and nonviral substrate analogs.

Sawyer TK, Staples DJ, Liu L, Tomasselli AG, Hui JO, O'Connell K, Schostarez H, Hester JB, Moon J, Howe WJ, et al. Sawyer TK, et al. Among authors: staples dj. Int J Pept Protein Res. 1992 Sep-Oct;40(3-4):274-81. doi: 10.1111/j.1399-3011.1992.tb00302.x. Int J Pept Protein Res. 1992. PMID: 1478785

5

Alpha-melanocyte stimulating hormone message and inhibitory sequences: comparative structure-activity studies on melanocytes.

Sawyer TK, Staples DJ, Castrucci AM, Hadley ME, al-Obeidi FA, Cody WL, Hruby VJ. Sawyer TK, et al. Among authors: staples dj. Peptides. 1990 Mar-Apr;11(2):351-7. doi: 10.1016/0196-9781(90)90092-j. Peptides. 1990. PMID: 2162535

6

Discovery and structure-activity relationships of novel alpha-melanocyte-stimulating hormone inhibitors.

Sawyer TK, Staples DJ, Castrucci AM, Hadley ME. Sawyer TK, et al. Among authors: staples dj. Pept Res. 1989 Jan-Feb;2(1):140-6. Pept Res. 1989. PMID: 2562482

7

Structure-conformation relationships of synthetic peptide inhibitors of human renin studied by resonance energy transfer and molecular modeling.

Epps DE, Mao B, Staples DJ, Sawyer TK. Epps DE, et al. Among authors: staples dj. Int J Pept Protein Res. 1988 Jan;31(1):22-34. doi: 10.1111/j.1399-3011.1988.tb00003.x. Int J Pept Protein Res. 1988. PMID: 3284834

8

Structure-activity relationships of [Nle4, D-Phe7]alpha-MSH. Discovery of a tripeptidyl agonist exhibiting sustained bioactivity.

Sawyer TK, Castrucci AM, Staples DJ, Affholter JA, De Vaux A, Hruby VJ, Hadley ME. Sawyer TK, et al. Among authors: staples dj. Ann N Y Acad Sci. 1993 May 31;680:597-9. doi: 10.1111/j.1749-6632.1993.tb19749.x. Ann N Y Acad Sci. 1993. PMID: 8390200 No abstract available.

9

Spectroscopic analysis of [Trp3]-beta-casomorphin analogs. Comparative structure conformation-activity studies.

Epps DE, Havel HA, Sawyer TK, Staples DJ, Chung NN, Schiller PW, Hartrodt B, Barth A. Epps DE, et al. Among authors: staples dj. Int J Pept Protein Res. 1991 Apr;37(4):257-67. doi: 10.1111/j.1399-3011.1991.tb00738.x. Int J Pept Protein Res. 1991. PMID: 1894441

10

Substrate analogue inhibition and active site titration of purified recombinant HIV-1 protease.

Tomasselli AG, Olsen MK, Hui JO, Staples DJ, Sawyer TK, Heinrikson RL, Tomich CS. Tomasselli AG, et al. Among authors: staples dj. Biochemistry. 1990 Jan 9;29(1):264-9. doi: 10.1021/bi00453a036. Biochemistry. 1990. PMID: 2182116

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

25 results

Search Page

Filters