Czarniecki MF - Search Results

1

Synthesis and structure-activity relationships of new disubstituted phenyl-containing 3,4-diamino-3-cyclobutene-1,2-diones as CXCR2 receptor antagonists.

Lai G, Merritt JR, He Z, Feng D, Chao J, Czarniecki MF, Rokosz LL, Stauffer TM, Rindgen D, Taveras AG. Lai G, et al. Among authors: czarniecki mf. Bioorg Med Chem Lett. 2008 Mar 15;18(6):1864-8. doi: 10.1016/j.bmcl.2008.02.010. Epub 2008 Feb 10. Bioorg Med Chem Lett. 2008. PMID: 18304809

2

T-type calcium channel blockers: spiro-piperidine azetidines and azetidinones-optimization, design and synthesis.

Smith EM, Sorota S, Kim HM, McKittrick BA, Nechuta TL, Bennett C, Knutson C, Burnett DA, Kieselgof J, Tan Z, Rindgen D, Bridal T, Zhou X, Jia YP, Dong Z, Mullins D, Zhang X, Priestley T, Correll CC, Tulshian D, Czarniecki M, Greenlee WJ. Smith EM, et al. Bioorg Med Chem Lett. 2010 Aug 1;20(15):4602-6. doi: 10.1016/j.bmcl.2010.06.012. Epub 2010 Jun 8. Bioorg Med Chem Lett. 2010. PMID: 20580233

3

Synthesis and SAR development of novel P2X7 receptor antagonists for the treatment of pain: part 2.

Brumfield S, Matasi JJ, Tulshian D, Czarniecki M, Greenlee W, Garlisi C, Qiu H, Devito K, Chen SC, Sun Y, Bertorelli R, Ansell J, Geiss W, Le VD, Martin GS, Vellekoop SA, Haber J, Allard ML. Brumfield S, et al. Bioorg Med Chem Lett. 2011 Dec 15;21(24):7287-90. doi: 10.1016/j.bmcl.2011.10.037. Epub 2011 Oct 21. Bioorg Med Chem Lett. 2011. PMID: 22078214

4

Discovery and synthesis of a novel series of quinoline-based thrombin receptor (PAR-1) antagonists.

Clasby MC, Chackalamannil S, Czarniecki M, Doller D, Eagen K, Greenlee WJ, Lin Y, Tsai H, Xia Y, Ahn HS, Agans-Fantuzzi J, Boykow G, Chintala M, Foster C, Bryant M, Lau J. Clasby MC, et al. Bioorg Med Chem Lett. 2006 Mar 15;16(6):1544-8. doi: 10.1016/j.bmcl.2005.12.042. Epub 2005 Dec 27. Bioorg Med Chem Lett. 2006. PMID: 16380251

5

Himbacine derived thrombin receptor antagonists: discovery of a new tricyclic core.

Clasby MC, Chackalamannil S, Czarniecki M, Doller D, Eagen K, Greenlee WJ, Lin Y, Tagat JR, Tsai H, Xia Y, Ahn HS, Agans-Fantuzzi J, Boykow G, Chintala M, Hsieh Y, McPhail AT. Clasby MC, et al. Bioorg Med Chem Lett. 2007 Jul 1;17(13):3647-51. doi: 10.1016/j.bmcl.2007.04.061. Epub 2007 Apr 25. Bioorg Med Chem Lett. 2007. PMID: 17490877

6

Structure-activity relationships of pyrroloquinazolines as thrombin receptor antagonists.

Ahn HS, Arik L, Boykow G, Burnett DA, Caplen MA, Czarniecki M, Domalski MS, Foster C, Manna M, Stamford AW, Wu Y. Ahn HS, et al. Bioorg Med Chem Lett. 1999 Jul 19;9(14):2073-8. doi: 10.1016/s0960-894x(99)00339-x. Bioorg Med Chem Lett. 1999. PMID: 10450984

7

Potent, low molecular weight thrombin receptor antagonists.

Chackalamannil S, Doller D, Eagen K, Czarniecki M, Ahn HS, Foster CJ, Boykow G. Chackalamannil S, et al. Bioorg Med Chem Lett. 2001 Nov 5;11(21):2851-3. doi: 10.1016/s0960-894x(01)00555-8. Bioorg Med Chem Lett. 2001. PMID: 11597414

8

Himbacine derived thrombin receptor (PAR-1) antagonists: structure-activity relationship of the lactone ring.

Xia Y, Chackalamannil S, Chan TM, Czarniecki M, Doller D, Eagen K, Greenlee WJ, Tsai H, Wang Y, Ahn HS, Boykow GC, McPhail AT. Xia Y, et al. Bioorg Med Chem Lett. 2006 Sep 15;16(18):4969-72. doi: 10.1016/j.bmcl.2006.06.042. Epub 2006 Jul 7. Bioorg Med Chem Lett. 2006. PMID: 16824760

9

Design, synthesis, and structure-activity relationship studies of himbacine derived muscarinic receptor antagonists.

Doller D, Chackalamannil S, Czarniecki M, McQuade R, Ruperto V. Doller D, et al. Bioorg Med Chem Lett. 1999 Mar 22;9(6):901-6. doi: 10.1016/s0960-894x(99)00101-8. Bioorg Med Chem Lett. 1999. PMID: 10206558

10

Design and discovery of 1,3-benzodiazepines as novel dopamine antagonists.

Zhu Z, Sun ZY, Ye Y, McKittrick B, Greenlee W, Czarniecki M, Fawzi A, Zhang H, Lachowicz JE. Zhu Z, et al. Bioorg Med Chem Lett. 2009 Sep 1;19(17):5218-21. doi: 10.1016/j.bmcl.2009.07.012. Epub 2009 Jul 9. Bioorg Med Chem Lett. 2009. PMID: 19643610

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