Piersanti G - Search Results

1

Switchable reactivity of acylated alpha, beta-dehydroamino ester in the Friedel-Crafts alkylation of indoles by changing the Lewis acid.

Angelini E, Balsamini C, Bartoccini F, Lucarini S, Piersanti G. Angelini E, et al. Among authors: piersanti g. J Org Chem. 2008 Jul 18;73(14):5654-7. doi: 10.1021/jo800881u. Epub 2008 Jun 18. J Org Chem. 2008. PMID: 18558761

2

2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.

Minetti P, Tinti MO, Carminati P, Castorina M, Di Cesare MA, Di Serio S, Gallo G, Ghirardi O, Giorgi F, Giorgi L, Piersanti G, Bartoccini F, Tarzia G. Minetti P, et al. Among authors: piersanti g. J Med Chem. 2005 Nov 3;48(22):6887-96. doi: 10.1021/jm058018d. J Med Chem. 2005. PMID: 16250647

3

Synthesis of benzo[1,2-d;3,4-d']diimidazole and 1H-pyrazolo[4,3-b]pyridine as putative A2A receptor antagonists.

Piersanti G, Giorgi L, Bartoccini F, Tarzia G, Minetti P, Gallo G, Giorgi F, Castorina M, Ghirardi O, Carminati P. Piersanti G, et al. Org Biomol Chem. 2007 Aug 21;5(16):2567-71. doi: 10.1039/b707599e. Org Biomol Chem. 2007. PMID: 18019530

4

An improved synthesis of cis-4-phenyl-2-propionamidotetralin (4-P-PDOT): a selective MT(2) melatonin receptor antagonist.

Lucarini S, Bedini A, Spadoni G, Piersanti G. Lucarini S, et al. Among authors: piersanti g. Org Biomol Chem. 2008 Jan 7;6(1):147-50. doi: 10.1039/b713904g. Epub 2007 Nov 13. Org Biomol Chem. 2008. PMID: 18075659

5

Direct preparation of unsymmetrical difunctionalized cyclen derivatives by an Ugi multicomponent reaction.

Piersanti G, Remi F, Fusi V, Formica M, Giorgi L, Zappia G. Piersanti G, et al. Org Lett. 2009 Jan 15;11(2):417-20. doi: 10.1021/ol802674r. Org Lett. 2009. PMID: 19090699

6

Diastereo- and enantioselective hydrogenation of a challenging enamide derived from 4-phenyl-2-tetralone: an appealing shortcut towards enantiopure cis-2-aminotetraline derivatives.

Lucarini S, Alessi M, Bedini A, Giorgini G, Piersanti G, Spadoni G. Lucarini S, et al. Among authors: piersanti g. Chem Asian J. 2010 Mar 1;5(3):550-4. doi: 10.1002/asia.200900441. Chem Asian J. 2010. PMID: 20108301

7

Direct B-alkyl Suzuki-Miyaura cross-coupling of 2-halopurines. Practical synthesis of ST1535, a potent adenosine A2A receptor antagonist.

Bartoccini F, Cabri W, Celona D, Minetti P, Piersanti G, Tarzia G. Bartoccini F, et al. Among authors: piersanti g. J Org Chem. 2010 Aug 6;75(15):5398-401. doi: 10.1021/jo101027h. J Org Chem. 2010. PMID: 20597521

8

A novel one-pot approach of hexahydropyrrolo[2,3-b]indole nucleus by a cascade addition/cyclization strategy: synthesis of (+/-)-esermethole.

Lucarini S, Bartoccini F, Battistoni F, Diamantini G, Piersanti G, Righi M, Spadoni G. Lucarini S, et al. Among authors: piersanti g. Org Lett. 2010 Sep 3;12(17):3844-7. doi: 10.1021/ol101527j. Org Lett. 2010. PMID: 20795744

9

Direct, one-pot reductive alkylation of anilines with functionalized acetals mediated by triethylsilane and TFA. Straightforward route for unsymmetrically substituted ethylenediamine.

Righi M, Bedini A, Piersanti G, Romagnoli F, Spadoni G. Righi M, et al. Among authors: piersanti g. J Org Chem. 2011 Jan 21;76(2):704-7. doi: 10.1021/jo102109f. Epub 2010 Dec 22. J Org Chem. 2011. PMID: 21175194

10

Synthesis and configuration determination of all enantiopure stereoisomers of the melatonin receptor ligand 4-phenyl-2-propionamidotetralin using an expedient optical resolution of 4-phenyl-2-tetralone.

Lucarini S, Bartolucci S, Bedini A, Gatti G, Orlando P, Piersanti G, Spadoni G. Lucarini S, et al. Among authors: piersanti g. Org Biomol Chem. 2012 Jan 14;10(2):305-13. doi: 10.1039/c1ob06369c. Epub 2011 Nov 18. Org Biomol Chem. 2012. PMID: 22095411

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