Kaatz GW - Search Results

1

From phenothiazine to 3-phenyl-1,4-benzothiazine derivatives as inhibitors of the Staphylococcus aureus NorA multidrug efflux pump.

Sabatini S, Kaatz GW, Rossolini GM, Brandini D, Fravolini A. Sabatini S, et al. Among authors: kaatz gw. J Med Chem. 2008 Jul 24;51(14):4321-30. doi: 10.1021/jm701623q. Epub 2008 Jun 25. J Med Chem. 2008. PMID: 18578473

2

From 6-aminoquinolone antibacterials to 6-amino-7-thiopyranopyridinylquinolone ethyl esters as inhibitors of Staphylococcus aureus multidrug efflux pumps.

Pieroni M, Dimovska M, Brincat JP, Sabatini S, Carosati E, Massari S, Kaatz GW, Fravolini A. Pieroni M, et al. Among authors: kaatz gw. J Med Chem. 2010 Jun 10;53(11):4466-80. doi: 10.1021/jm1003304. J Med Chem. 2010. PMID: 20446747

3

Discovery of novel inhibitors of the NorA multidrug transporter of Staphylococcus aureus.

Brincat JP, Carosati E, Sabatini S, Manfroni G, Fravolini A, Raygada JL, Patel D, Kaatz GW, Cruciani G. Brincat JP, et al. Among authors: kaatz gw. J Med Chem. 2011 Jan 13;54(1):354-65. doi: 10.1021/jm1011963. Epub 2010 Dec 8. J Med Chem. 2011. PMID: 21141825

4

Evolution from a natural flavones nucleus to obtain 2-(4-Propoxyphenyl)quinoline derivatives as potent inhibitors of the S. aureus NorA efflux pump.

Sabatini S, Gosetto F, Manfroni G, Tabarrini O, Kaatz GW, Patel D, Cecchetti V. Sabatini S, et al. Among authors: kaatz gw. J Med Chem. 2011 Aug 25;54(16):5722-36. doi: 10.1021/jm200370y. Epub 2011 Aug 3. J Med Chem. 2011. PMID: 21751791

5

Pyrazolo[4,3-c][1,2]benzothiazines 5,5-dioxide: a promising new class of Staphylococcus aureus NorA efflux pump inhibitors.

Sabatini S, Gosetto F, Serritella S, Manfroni G, Tabarrini O, Iraci N, Brincat JP, Carosati E, Villarini M, Kaatz GW, Cecchetti V. Sabatini S, et al. Among authors: kaatz gw. J Med Chem. 2012 Apr 12;55(7):3568-72. doi: 10.1021/jm201446h. Epub 2012 Apr 3. J Med Chem. 2012. PMID: 22432682

6

Re-evolution of the 2-phenylquinolines: ligand-based design, synthesis, and biological evaluation of a potent new class of Staphylococcus aureus NorA efflux pump inhibitors to combat antimicrobial resistance.

Sabatini S, Gosetto F, Iraci N, Barreca ML, Massari S, Sancineto L, Manfroni G, Tabarrini O, Dimovska M, Kaatz GW, Cecchetti V. Sabatini S, et al. Among authors: kaatz gw. J Med Chem. 2013 Jun 27;56(12):4975-89. doi: 10.1021/jm400262a. Epub 2013 Jun 13. J Med Chem. 2013. PMID: 23710549

7

Ligand Promiscuity between the Efflux Pumps Human P-Glycoprotein and S. aureus NorA.

Brincat JP, Broccatelli F, Sabatini S, Frosini M, Neri A, Kaatz GW, Cruciani G, Carosati E. Brincat JP, et al. Among authors: kaatz gw. ACS Med Chem Lett. 2012 Jan 23;3(3):248-51. doi: 10.1021/ml200293c. eCollection 2012 Mar 8. ACS Med Chem Lett. 2012. PMID: 24900460 Free PMC article.

8

Pharmacophore-Based Repositioning of Approved Drugs as Novel Staphylococcus aureus NorA Efflux Pump Inhibitors.

Astolfi A, Felicetti T, Iraci N, Manfroni G, Massari S, Pietrella D, Tabarrini O, Kaatz GW, Barreca ML, Sabatini S, Cecchetti V. Astolfi A, et al. Among authors: kaatz gw. J Med Chem. 2017 Feb 23;60(4):1598-1604. doi: 10.1021/acs.jmedchem.6b01439. Epub 2017 Feb 8. J Med Chem. 2017. PMID: 28117588

9

Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3-Phenyl-1,4-benzothiazine Analogues.

Felicetti T, Cannalire R, Burali MS, Massari S, Manfroni G, Barreca ML, Tabarrini O, Schindler BD, Sabatini S, Kaatz GW, Cecchetti V. Felicetti T, et al. Among authors: kaatz gw. ChemMedChem. 2017 Aug 22;12(16):1293-1302. doi: 10.1002/cmdc.201700286. Epub 2017 Jul 17. ChemMedChem. 2017. PMID: 28598572

10

Studies on 2-phenylquinoline Staphylococcus aureus NorA efflux pump inhibitors: New insights on the C-6 position.

Felicetti T, Cannalire R, Nizi MG, Tabarrini O, Massari S, Barreca ML, Manfroni G, Schindler BD, Cecchetti V, Kaatz GW, Sabatini S. Felicetti T, et al. Among authors: kaatz gw. Eur J Med Chem. 2018 Jul 15;155:428-433. doi: 10.1016/j.ejmech.2018.06.013. Epub 2018 Jun 6. Eur J Med Chem. 2018. PMID: 29908437

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

130 results

Search Page

Filters