Vassiliou S - Search Results

1

Design, synthesis, and evaluation of novel organophosphorus inhibitors of bacterial ureases.

Vassiliou S, Grabowiecka A, Kosikowska P, Yiotakis A, Kafarski P, Berlicki Ł. Vassiliou S, et al. J Med Chem. 2008 Sep 25;51(18):5736-44. doi: 10.1021/jm800570q. Epub 2008 Aug 22. J Med Chem. 2008. PMID: 18717581

2

Computer-aided optimization of phosphinic inhibitors of bacterial ureases.

Vassiliou S, Kosikowska P, Grabowiecka A, Yiotakis A, Kafarski P, Berlicki L. Vassiliou S, et al. J Med Chem. 2010 Aug 12;53(15):5597-606. doi: 10.1021/jm100340m. J Med Chem. 2010. PMID: 20684601

3

Novel organophosphorus scaffolds of urease inhibitors obtained by substitution of Morita-Baylis-Hillman adducts with phosphorus nucleophiles.

Ntatsopoulos V, Vassiliou S, Macegoniuk K, Berlicki Ł, Mucha A. Ntatsopoulos V, et al. Among authors: vassiliou s. Eur J Med Chem. 2017 Jun 16;133:107-120. doi: 10.1016/j.ejmech.2017.03.070. Epub 2017 Mar 29. Eur J Med Chem. 2017. PMID: 28384543

4

Structural exploration of cinnamate-based phosphonic acids as inhibitors of bacterial ureases.

Ntatsopoulos V, Macegoniuk K, Mucha A, Vassiliou S, Berlicki Ł. Ntatsopoulos V, et al. Among authors: vassiliou s. Eur J Med Chem. 2018 Nov 5;159:307-316. doi: 10.1016/j.ejmech.2018.09.074. Epub 2018 Oct 2. Eur J Med Chem. 2018. PMID: 30300843

5

Catechol-based inhibitors of bacterial urease.

Pagoni A, Daliani T, Macegoniuk K, Vassiliou S, Berlicki Ł. Pagoni A, et al. Among authors: vassiliou s. Bioorg Med Chem Lett. 2019 May 1;29(9):1085-1089. doi: 10.1016/j.bmcl.2019.02.032. Epub 2019 Feb 27. Bioorg Med Chem Lett. 2019. PMID: 30850166

6

Covalent Inhibition of Bacterial Urease by Bifunctional Catechol-Based Phosphonates and Phosphinates.

Pagoni A, Grabowiecka A, Tabor W, Mucha A, Vassiliou S, Berlicki Ł. Pagoni A, et al. Among authors: vassiliou s. J Med Chem. 2021 Jan 14;64(1):404-416. doi: 10.1021/acs.jmedchem.0c01143. Epub 2020 Dec 28. J Med Chem. 2021. PMID: 33369409

7

A synthetic method for diversification of the P1' substituent in phosphinic dipeptides as a tool for exploration of the specificity of the S1' binding pockets of leucine aminopeptidases.

Vassiliou S, Xeilari M, Yiotakis A, Grembecka J, Pawełczak M, Kafarski P, Mucha A. Vassiliou S, et al. Bioorg Med Chem. 2007 May 1;15(9):3187-200. doi: 10.1016/j.bmc.2007.02.042. Epub 2007 Feb 22. Bioorg Med Chem. 2007. PMID: 17337192

8

Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases.

Vassiliou S, Węglarz-Tomczak E, Berlicki Ł, Pawełczak M, Nocek B, Mulligan R, Joachimiak A, Mucha A. Vassiliou S, et al. J Med Chem. 2014 Oct 9;57(19):8140-51. doi: 10.1021/jm501071f. Epub 2014 Sep 22. J Med Chem. 2014. PMID: 25192493 Free PMC article.

9

Cyclic peptides with a phosphinic bond as potent inhibitors of a zinc bacterial collagenase.

Yiotakis A, Lecoq A, Vassiliou S, Raynal I, Cuniasse P, Dive V. Yiotakis A, et al. Among authors: vassiliou s. J Med Chem. 1994 Aug 19;37(17):2713-20. doi: 10.1021/jm00043a011. J Med Chem. 1994. PMID: 8064799

10

Phosphinic pseudo-tripeptides as potent inhibitors of matrix metalloproteinases: a structure-activity study.

Vassiliou S, Mucha A, Cuniasse P, Georgiadis D, Lucet-Levannier K, Beau F, Kannan R, Murphy G, Knäuper V, Rio MC, Basset P, Yiotakis A, Dive V. Vassiliou S, et al. J Med Chem. 1999 Jul 15;42(14):2610-20. doi: 10.1021/jm9900164. J Med Chem. 1999. PMID: 10411481

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