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Page 1
Discovery of orally bioavailable cathepsin S inhibitors for the reversal of neuropathic pain.
Irie O, Kosaka T, Ehara T, Yokokawa F, Kanazawa T, Hirao H, Iwasaki A, Sakaki J, Teno N, Hitomi Y, Iwasaki G, Fukaya H, Nonomura K, Tanabe K, Koizumi S, Uchiyama N, Bevan SJ, Malcangio M, Gentry C, Fox AJ, Yaqoob M, Culshaw AJ, Allan Hallett. Irie O, et al. Among authors: malcangio m. J Med Chem. 2008 Sep 25;51(18):5502-5. doi: 10.1021/jm800839j. J Med Chem. 2008. PMID: 18754655
Overcoming hERG issues for brain-penetrating cathepsin S inhibitors: 2-cyanopyrimidines. Part 2.
Irie O, Kosaka T, Kishida M, Sakaki J, Masuya K, Konishi K, Yokokawa F, Ehara T, Iwasaki A, Iwaki Y, Hitomi Y, Toyao A, Gunji H, Teno N, Iwasaki G, Hirao H, Kanazawa T, Tanabe K, Hiestand PC, Malcangio M, Fox AJ, Bevan SJ, Yaqoob M, Culshaw AJ, Hart TW, Hallett A. Irie O, et al. Among authors: malcangio m. Bioorg Med Chem Lett. 2008 Oct 1;18(19):5280-4. doi: 10.1016/j.bmcl.2008.08.067. Epub 2008 Aug 22. Bioorg Med Chem Lett. 2008. PMID: 18783943
Role of the cysteine protease cathepsin S in neuropathic hyperalgesia.
Barclay J, Clark AK, Ganju P, Gentry C, Patel S, Wotherspoon G, Buxton F, Song C, Ullah J, Winter J, Fox A, Bevan S, Malcangio M. Barclay J, et al. Among authors: malcangio m. Pain. 2007 Aug;130(3):225-234. doi: 10.1016/j.pain.2006.11.017. Epub 2007 Jan 23. Pain. 2007. PMID: 17250968
Inhibition of spinal microglial cathepsin S for the reversal of neuropathic pain.
Clark AK, Yip PK, Grist J, Gentry C, Staniland AA, Marchand F, Dehvari M, Wotherspoon G, Winter J, Ullah J, Bevan S, Malcangio M. Clark AK, et al. Among authors: malcangio m. Proc Natl Acad Sci U S A. 2007 Jun 19;104(25):10655-60. doi: 10.1073/pnas.0610811104. Epub 2007 Jun 5. Proc Natl Acad Sci U S A. 2007. PMID: 17551020 Free PMC article.
A distinct role for transient receptor potential ankyrin 1, in addition to transient receptor potential vanilloid 1, in tumor necrosis factor α-induced inflammatory hyperalgesia and Freund's complete adjuvant-induced monarthritis.
Fernandes ES, Russell FA, Spina D, McDougall JJ, Graepel R, Gentry C, Staniland AA, Mountford DM, Keeble JE, Malcangio M, Bevan S, Brain SD. Fernandes ES, et al. Among authors: malcangio m. Arthritis Rheum. 2011 Mar;63(3):819-29. doi: 10.1002/art.30150. Arthritis Rheum. 2011. PMID: 21360511 Free article.
Environmental cold exposure increases blood flow and affects pain sensitivity in the knee joints of CFA-induced arthritic mice in a TRPA1-dependent manner.
Fernandes ES, Russell FA, Alawi KM, Sand C, Liang L, Salamon R, Bodkin JV, Aubdool AA, Arno M, Gentry C, Smillie SJ, Bevan S, Keeble JE, Malcangio M, Brain SD. Fernandes ES, et al. Among authors: malcangio m. Arthritis Res Ther. 2016 Jan 11;18:7. doi: 10.1186/s13075-015-0905-x. Arthritis Res Ther. 2016. PMID: 26754745 Free PMC article.
136 results