Gilbert AM - Search Results

1

N-((8-hydroxy-5-substituted-quinolin-7-yl)(phenyl)methyl)-2-phenyloxy/amino-acetamide inhibitors of ADAMTS-5 (Aggrecanase-2).

Gilbert AM, Bursavich MG, Lombardi S, Georgiadis KE, Reifenberg E, Flannery CR, Morris EA. Gilbert AM, et al. Bioorg Med Chem Lett. 2008 Dec 15;18(24):6454-7. doi: 10.1016/j.bmcl.2008.10.065. Epub 2008 Oct 18. Bioorg Med Chem Lett. 2008. PMID: 18974001

2

Design and SAR of novel potassium channel openers targeted for urge urinary incontinence. 2. Selective and potent benzylamino cyclobutenediones.

Gilbert AM, Antane MM, Argentieri TM, Butera JA, Francisco GD, Freeden C, Gundersen EG, Graceffa RF, Herbst D, Hirth BH, Lennox JR, McFarlane G, Norton NW, Quagliato D, Sheldon JH, Warga D, Wojdan A, Woods M. Gilbert AM, et al. J Med Chem. 2000 Mar 23;43(6):1203-14. doi: 10.1021/jm9905108. J Med Chem. 2000. PMID: 10737753

3

Novel and selective calcitonin-inducing agents.

Gilbert AM, Caltabiano S, Roberts D, Sum SF, Francisco GD, Lim K, Asselin M, Ellingboe JW, Kharode Y, Cannistraci A, Francis R, TrailSmith M, Gralnick D. Gilbert AM, et al. J Med Chem. 2000 Mar 23;43(6):1223-33. doi: 10.1021/jm990558l. J Med Chem. 2000. PMID: 10737755

4

Pyrazolopyrimidine-2,4-dione sulfonamides: novel and selective calcitonin inducers.

Gilbert AM, Caltabiano S, Koehn FE, Chen ZJ, Francisco GD, Ellingboe JW, Kharode Y, Mangine A, Francis R, TrailSmith M, Gralnick D. Gilbert AM, et al. J Med Chem. 2002 May 23;45(11):2342-5. doi: 10.1021/jm010554s. J Med Chem. 2002. PMID: 12014973

5

Anthranilate 4H-oxazol-5-ones: novel small molecule antibacterial acyl carrier protein synthase (AcpS) inhibitors.

Gilbert AM, Kirisits M, Toy P, Nunn DS, Failli A, Dushin EG, Novikova E, Petersen PJ, Joseph-McCarthy D, McFadyen I, Fritz CC. Gilbert AM, et al. Bioorg Med Chem Lett. 2004 Jan 5;14(1):37-41. doi: 10.1016/j.bmcl.2003.10.032. Bioorg Med Chem Lett. 2004. PMID: 14684293

6

Modulation of selective serotonin reuptake inhibitor and 5-HT1A antagonist activity in 8-aza-bicyclo[3.2.1]octane derivatives of 2,3-dihydro-1,4-benzodioxane.

Gilbert AM, Stack GP, Nilakantan R, Kodah J, Tran M, Scerni R, Shi X, Smith DL, Andree TH. Gilbert AM, et al. Bioorg Med Chem Lett. 2004 Jan 19;14(2):515-8. doi: 10.1016/j.bmcl.2003.10.024. Bioorg Med Chem Lett. 2004. PMID: 14698193

7

Novel aryloxy-8-azabicyclo[3.2.1]oct-3-enes with 5-HT transporter and 5-HT1A affinity.

Gilbert AM, Coleman T, Kodah J, Mewshaw RE, Scerni R, Schechter LE, Smith DL, Andree TH. Gilbert AM, et al. Bioorg Med Chem Lett. 2004 Nov 1;14(21):5281-4. doi: 10.1016/j.bmcl.2004.08.030. Bioorg Med Chem Lett. 2004. PMID: 15454211

8

Expedient parallel synthesis of 2-amino-4-heteroarylpyrimidines.

Bursavich MG, Lombardi S, Gilbert AM. Bursavich MG, et al. Among authors: gilbert am. Org Lett. 2005 Sep 15;7(19):4113-6. doi: 10.1021/ol051339z. Org Lett. 2005. PMID: 16146365

9

Pyrazolidine-3,5-diones and 5-hydroxy-1H-pyrazol-3(2H)-ones, inhibitors of UDP-N-acetylenolpyruvyl glucosamine reductase.

Gilbert AM, Failli A, Shumsky J, Yang Y, Severin A, Singh G, Hu W, Keeney D, Petersen PJ, Katz AH. Gilbert AM, et al. J Med Chem. 2006 Oct 5;49(20):6027-36. doi: 10.1021/jm060499t. J Med Chem. 2006. PMID: 17004716

10

Synthesis and evaluation of aryl thioxothiazolidinone inhibitors of ADAMTS-5 (Aggrecanase-2).

Bursavich MG, Gilbert AM, Lombardi S, Georgiadis KE, Reifenberg E, Flannery CR, Morris EA. Bursavich MG, et al. Among authors: gilbert am. Bioorg Med Chem Lett. 2007 Mar 1;17(5):1185-8. doi: 10.1016/j.bmcl.2006.12.027. Epub 2006 Dec 12. Bioorg Med Chem Lett. 2007. PMID: 17210251

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

71 results

Search Page

Filters