Kikelj D - Search Results

1

Synthesis and biological evaluation of new glutamic acid-based inhibitors of MurD ligase.

Tomasić T, Zidar N, Rupnik V, Kovac A, Blanot D, Gobec S, Kikelj D, Masic LP. Tomasić T, et al. Among authors: kikelj d. Bioorg Med Chem Lett. 2009 Jan 1;19(1):153-7. doi: 10.1016/j.bmcl.2008.10.129. Epub 2008 Nov 5. Bioorg Med Chem Lett. 2009. PMID: 19014883

2

N-[trans-2-[[2'-(acetylamino)cyclohexyl]oxy]acetyl]-L-alanyl-D-glutamic acid: a novel immunologically active carbocyclic muramyl dipeptide analogue.

Kikelj D, Pecar S, Kotnik V, Stalc A, Wraber-Herzog B, Simcic S, Ihan A, Klamfer L, Povsic L, Grahek R, Suhadolc E, Hocevar M, Hönig H, Rogi-Kohlenprath R. Kikelj D, et al. J Med Chem. 1998 Feb 12;41(4):530-9. doi: 10.1021/jm970509d. J Med Chem. 1998. PMID: 9484503

3

Design and structure-activity relationship of thrombin inhibitors with an azaphenylalanine scaffold: potency and selectivity enhancements via P2 optimization.

Zega A, Mlinsek G, Sepic P, Golic Grdadolnik S, Solmajer T, Tschopp TB, Steiner B, Kikelj D, Urleb U. Zega A, et al. Among authors: kikelj d. Bioorg Med Chem. 2001 Oct;9(10):2745-56. doi: 10.1016/s0968-0896(01)00202-4. Bioorg Med Chem. 2001. PMID: 11557360

4

Novel thrombin inhibitors incorporating non-basic partially saturated heterobicyclic P1-arginine mimetics.

Peterlin-Masic L, Mlinsek G, Solmajer T, Trampus-Bakija A, Stegnar M, Kikelj D. Peterlin-Masic L, et al. Among authors: kikelj d. Bioorg Med Chem Lett. 2003 Mar 10;13(5):789-94. doi: 10.1016/s0960-894x(03)00030-1. Bioorg Med Chem Lett. 2003. PMID: 12617892

5

Selective 3-amino-2-pyridinone acetamide thrombin inhibitors incorporating weakly basic partially saturated heterobicyclic P1-arginine mimetics.

Peterlin-Masic L, Kranjc A, Marinko P, Mlinsek G, Solmajer T, Stegnar M, Kikelj D. Peterlin-Masic L, et al. Among authors: kikelj d. Bioorg Med Chem Lett. 2003 Oct 6;13(19):3171-6. doi: 10.1016/s0960-894x(03)00717-0. Bioorg Med Chem Lett. 2003. PMID: 12951087

6

Novel thrombin inhibitors incorporating weakly basic heterobicyclic P1-arginine mimetics: optimization via modification of P1 and P3 moieties.

Kranjc A, Peterlin-Masic L, Ilas J, Prezelj A, Stegnar M, Kikelj D. Kranjc A, et al. Among authors: kikelj d. Bioorg Med Chem Lett. 2004 Jun 21;14(12):3251-6. doi: 10.1016/j.bmcl.2004.03.085. Bioorg Med Chem Lett. 2004. PMID: 15149685

7

Phosphonate inhibitors of antigen 85C, a crucial enzyme involved in the biosynthesis of the Mycobacterium tuberculosis cell wall.

Gobec S, Plantan I, Mravljak J, Wilson RA, Besra GS, Kikelj D. Gobec S, et al. Among authors: kikelj d. Bioorg Med Chem Lett. 2004 Jul 5;14(13):3559-62. doi: 10.1016/j.bmcl.2004.04.052. Bioorg Med Chem Lett. 2004. PMID: 15177473

8

Toward a novel class of antithrombotic compounds with dual function. Discovery of 1,4-benzoxazin-3(4H)-one derivatives possessing thrombin inhibitory and fibrinogen receptor antagonistic activities.

Stefanic Anderluh P, Anderluh M, Ilas J, Mravljak J, Sollner Dolenc M, Stegnar M, Kikelj D. Stefanic Anderluh P, et al. Among authors: kikelj d. J Med Chem. 2005 May 5;48(9):3110-3. doi: 10.1021/jm048984g. J Med Chem. 2005. PMID: 15857114

9

Novel pyrazinone and pyridinone thrombin inhibitors incorporating weakly basic heterobicyclic P(1)-arginine mimetics.

Kranjc A, Masic LP, Reven S, Mikic K, Prezelj A, Stegnar M, Kikelj D. Kranjc A, et al. Among authors: kikelj d. Eur J Med Chem. 2005 Aug;40(8):782-91. doi: 10.1016/j.ejmech.2005.03.007. Eur J Med Chem. 2005. PMID: 15890436

10

Design, synthesis, biochemical evaluation and antimycobacterial action of phosphonate inhibitors of antigen 85C, a crucial enzyme involved in biosynthesis of the mycobacterial cell wall.

Gobec S, Plantan I, Mravljak J, Svajger U, Wilson RA, Besra GS, Soares SL, Appelberg R, Kikelj D. Gobec S, et al. Among authors: kikelj d. Eur J Med Chem. 2007 Jan;42(1):54-63. doi: 10.1016/j.ejmech.2006.08.007. Epub 2006 Sep 28. Eur J Med Chem. 2007. PMID: 17010479

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