Kowal D - Search Results

1

Prodrugs of perzinfotel with improved oral bioavailability.

Baudy RB, Butera JA, Abou-Gharbia MA, Chen H, Harrison B, Jain U, Magolda R, Sze JY, Brandt MR, Cummons TA, Kowal D, Pangalos MN, Zupan B, Hoffmann M, May M, Mugford C, Kennedy J, Childers WE Jr. Baudy RB, et al. Among authors: kowal d. J Med Chem. 2009 Feb 12;52(3):771-8. doi: 10.1021/jm8011799. J Med Chem. 2009. PMID: 19146418

2

Design, synthesis, SAR, and biological evaluation of highly potent benzimidazole-spaced phosphono-alpha-amino acid competitive NMDA antagonists of the AP-6 type.

Baudy RB, Fletcher H 3rd, Yardley JP, Zaleska MM, Bramlett DR, Tasse RP, Kowal DM, Katz AH, Moyer JA, Abou-Gharbia M. Baudy RB, et al. Among authors: kowal dm. J Med Chem. 2001 May 10;44(10):1516-29. doi: 10.1021/jm000385w. J Med Chem. 2001. PMID: 11334562

3

Potent quinoxaline-spaced phosphono alpha-amino acids of the AP-6 type as competitive NMDA antagonists: synthesis and biological evaluation.

Baudy RB, Greenblatt LP, Jirkovsky IL, Conklin M, Russo RJ, Bramlett DR, Emrey TA, Simmonds JT, Kowal DM, Stein RP, et al. Baudy RB, et al. Among authors: kowal dm. J Med Chem. 1993 Feb 5;36(3):331-42. doi: 10.1021/jm00055a004. J Med Chem. 1993. PMID: 8093907

4

Design and synthesis of [2-(8,9-dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl)-ethyl]phosphonic acid (EAA-090), a potent N-methyl-D-aspartate antagonist, via the use of 3-cyclobutene-1,2-dione as an achiral alpha-amino acid bioisostere.

Kinney WA, Abou-Gharbia M, Garrison DT, Schmid J, Kowal DM, Bramlett DR, Miller TL, Tasse RP, Zaleska MM, Moyer JA. Kinney WA, et al. Among authors: kowal dm. J Med Chem. 1998 Jan 15;41(2):236-46. doi: 10.1021/jm970504g. J Med Chem. 1998. PMID: 9457246

5

Bioisosteric replacement of the alpha-amino carboxylic acid functionality in 2-amino-5-phosphonopentanoic acid yields unique 3,4-diamino-3-cyclobutene-1,2-dione containing NMDA antagonists.

Kinney WA, Lee NE, Garrison DT, Podlesny EJ Jr, Simmonds JT, Bramlett D, Notvest RR, Kowal DM, Tasse RP. Kinney WA, et al. Among authors: kowal dm. J Med Chem. 1992 Dec 11;35(25):4720-6. doi: 10.1021/jm00103a010. J Med Chem. 1992. PMID: 1361582

6

A [35S]GTPgammaS binding assessment of metabotropic glutamate receptor standards in Chinese hamster ovary cell lines expressing the human metabotropic receptor subtypes 2 and 4.

Kowal D, Hsiao CL, Ge A, Wardwell-Swanson J, Ghosh K, Tasse R. Kowal D, et al. Neuropharmacology. 1998;37(2):179-87. doi: 10.1016/s0028-3908(98)00011-2. Neuropharmacology. 1998. PMID: 9680242

7

Design and models for estimating antagonist potency (pA2, Kd and IC50) following the detection of antagonism observed in the presence of intrinsic activity.

Ghosh K, Kowal D, Dawson LA, Tasse R. Ghosh K, et al. Among authors: kowal d. Neuropharmacology. 1999 Mar;38(3):361-73. doi: 10.1016/s0028-3908(98)00185-3. Neuropharmacology. 1999. PMID: 10219974

8

The effect of conjugated equine estrogens on ovariectomy-induced osteopenia in the rat.

Hayward MA, Kharode YP, Becci MM, Kowal D. Hayward MA, et al. Among authors: kowal d. Agents Actions. 1990 Aug;31(1-2):152-6. doi: 10.1007/BF02003236. Agents Actions. 1990. PMID: 2178316

9

Smartphone App-Based Remote Monitoring Challenges in Patients with Cardiac Resynchronization Therapy Defibrillators-A Multicenter Study.

Kowal D, Prech M, Katarzyńska-Szymańska A, Baszko A, Skonieczny G, Wabich E, Kempa M, Rubiś B, Mitkowski P. Kowal D, et al. J Clin Med. 2024 Oct 23;13(21):6323. doi: 10.3390/jcm13216323. J Clin Med. 2024. PMID: 39518463 Free PMC article.

10

Spatial Variability in Relationships between Early Childhood Lead Exposure and Standardized Test Scores in Fourth Grade North Carolina Public School Students (2013-2016).

Bravo MA, Kowal DR, Zephyr D, Feldman J, Ensor K, Miranda ML. Bravo MA, et al. Among authors: kowal dr. Environ Health Perspect. 2024 Sep;132(9):97003. doi: 10.1289/EHP13898. Epub 2024 Sep 3. Environ Health Perspect. 2024. PMID: 39226183 Free PMC article.

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