Summa V - Search Results

1

Structural characterization of the Hepatitis C Virus NS3 protease from genotype 3a: the basis of the genotype 1b vs. 3a inhibitor potency shift.

Gallo M, Bottomley MJ, Pennestri M, Eliseo T, Paci M, Koch U, Bazzo R, Summa V, Carfì A, Cicero DO. Gallo M, et al. Among authors: summa v. Virology. 2010 Sep 30;405(2):424-38. doi: 10.1016/j.virol.2010.05.035. Epub 2010 Jul 13. Virology. 2010. PMID: 20630554 Free article.

2

Optimization of Ursolic Acid Extraction in Oil from Annurca Apple to Obtain Oleolytes with Potential Cosmeceutical Application.

Maisto M, Piccolo V, Novellino E, Schiano E, Iannuzzo F, Ciampaglia R, Summa V, Tenore GC. Maisto M, et al. Among authors: summa v. Antioxidants (Basel). 2023 Jan 18;12(2):224. doi: 10.3390/antiox12020224. Antioxidants (Basel). 2023. PMID: 36829781 Free PMC article.

3

Discovery of alpha,gamma-diketo acids as potent selective and reversible inhibitors of hepatitis C virus NS5b RNA-dependent RNA polymerase.

Summa V, Petrocchi A, Pace P, Matassa VG, De Francesco R, Altamura S, Tomei L, Koch U, Neuner P. Summa V, et al. J Med Chem. 2004 Jan 1;47(1):14-7. doi: 10.1021/jm0342109. J Med Chem. 2004. PMID: 14695815

4

From dihydroxypyrimidine carboxylic acids to carboxamide HIV-1 integrase inhibitors: SAR around the amide moiety.

Petrocchi A, Koch U, Matassa VG, Pacini B, Stillmock KA, Summa V. Petrocchi A, et al. Among authors: summa v. Bioorg Med Chem Lett. 2007 Jan 15;17(2):350-3. doi: 10.1016/j.bmcl.2006.10.054. Epub 2006 Oct 25. Bioorg Med Chem Lett. 2007. PMID: 17107799

5

Binding of a noncovalent inhibitor exploiting the S' region stabilizes the hepatitis C virus NS3 protease conformation in the absence of cofactor.

Gallo M, Pennestri M, Bottomley MJ, Barbato G, Eliseo T, Paci M, Narjes F, De Francesco R, Summa V, Koch U, Bazzo R, Cicero DO. Gallo M, et al. Among authors: summa v. J Mol Biol. 2009 Jan 30;385(4):1142-55. doi: 10.1016/j.jmb.2008.11.017. Epub 2008 Nov 24. J Mol Biol. 2009. PMID: 19061898

6

Inhibitors of hepatitis C virus NS3/4A: alpha-ketoamide based macrocyclic inhibitors.

Avolio S, Robertson K, Hernando JI, DiMuzio J, Summa V. Avolio S, et al. Among authors: summa v. Bioorg Med Chem Lett. 2009 Apr 15;19(8):2295-8. doi: 10.1016/j.bmcl.2009.02.079. Epub 2009 Feb 25. Bioorg Med Chem Lett. 2009. PMID: 19285390

7

Phosphorous acid analogs of novel P2-P4 macrocycles as inhibitors of HCV-NS3 protease.

Pompei M, Francesco ME, Koch U, Liverton NJ, Summa V. Pompei M, et al. Among authors: summa v. Bioorg Med Chem Lett. 2009 May 1;19(9):2574-8. doi: 10.1016/j.bmcl.2009.03.038. Epub 2009 Mar 17. Bioorg Med Chem Lett. 2009. PMID: 19328685

8

Inhibitors of the hepatitis C virus NS3 protease with basic amine functionality at the P3-amino acid N-terminus: discovery and optimization of a new series of P2-P4 macrocycles.

Harper S, Ferrara M, Crescenzi B, Pompei M, Palumbi MC, DiMuzio JM, Donghi M, Fiore F, Koch U, Liverton NJ, Pesci S, Petrocchi A, Rowley M, Summa V, Gardelli C. Harper S, et al. Among authors: summa v. J Med Chem. 2009 Aug 13;52(15):4820-37. doi: 10.1021/jm900372w. J Med Chem. 2009. PMID: 19624135

9

Novel macrocyclic inhibitors of hepatitis C NS3/4A protease featuring a 2-amino-1,3-thiazole as a P4 carbamate replacement.

Di Francesco ME, Dessole G, Nizi E, Pace P, Koch U, Fiore F, Pesci S, Di Muzio J, Monteagudo E, Rowley M, Summa V. Di Francesco ME, et al. Among authors: summa v. J Med Chem. 2009 Nov 26;52(22):7014-28. doi: 10.1021/jm900524b. J Med Chem. 2009. PMID: 19856919

10

Identification and biological evaluation of a series of 1H-benzo[de]isoquinoline-1,3(2H)-diones as hepatitis C virus NS5B polymerase inhibitors.

Ontoria JM, Rydberg EH, Di Marco S, Tomei L, Attenni B, Malancona S, Martin Hernando JI, Gennari N, Koch U, Narjes F, Rowley M, Summa V, Carroll SS, Olsen DB, De Francesco R, Altamura S, Migliaccio G, Carfì A. Ontoria JM, et al. Among authors: summa v. J Med Chem. 2009 Aug 27;52(16):5217-27. doi: 10.1021/jm900517t. J Med Chem. 2009. PMID: 19877603

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